Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50031663
TargetBeta-secretase 1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50316864([(2R,4S,5S)-5-(N-Boc-L-leucyl-L-phenylalanylamido)...)
Affinity DataIC50: 2.31E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50316861(N-((S)-1-((4S,5S,7R)-5-hydroxy-8-(isobutylamino)-2...)
Affinity DataIC50: 2.64E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50316860((2R,4S,5S)-4-hydroxy-N-isobutyl-2,7-dimethyl-5-((S...)
Affinity DataIC50: 3.79E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50316862(N-((S)-1-((4S,5S,7R)-5-hydroxy-8-(isobutylamino)-2...)
Affinity DataIC50: 3.81E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50316863(2,4-dichloro-N-((S)-1-((4S,5S,7R)-5-hydroxy-8-(iso...)
Affinity DataIC50: 4.24E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50316867(N-((S)-1-((4S,5S,7R)-5-hydroxy-8-(isobutylamino)-2...)
Affinity DataIC50: 4.67E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50316865(N-((S)-1-((4S,5S,7R)-5-hydroxy-8-(isobutylamino)-2...)
Affinity DataIC50: 6.93E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50316858(N-((S)-1-((4S,5S,7R)-5-hydroxy-8-(isobutylamino)-2...)
Affinity DataIC50: 8.07E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50316866(N-((S)-1-((4S,5S,7R)-5-hydroxy-8-(isobutylamino)-2...)
Affinity DataIC50: 1.57E+4nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50316859([(2R,4S,5S)-5-[N-(4-trifluoromethyl)benzoyl-L-phen...)
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed