Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50031121
TargetProteasome subunit beta type-5(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50: 1nMAssay Description:Inhibition of 26S proteasome beta 5 using LLVY as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307482((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50: 2nMAssay Description:Inhibition of 26S proteasome beta 5 using LLVY as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307480(Pyrazine-2-carboxylic acid(1-[3-methyl-1-(2,9,9-tr...)
Affinity DataIC50: 3nMAssay Description:Inhibition of 26S proteasome beta 5 using LLVY as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307479(Pyrazine-2-carboxylic acid(1-[3-methyl-1-(2,9,9-tr...)
Affinity DataIC50: 31nMAssay Description:Inhibition of 26S proteasome beta 5 using LLVY as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307483((S)-2-azido-N-((S)-1-((S)-3-(3,5-bis(trifluorometh...)
Affinity DataIC50: 100nMAssay Description:Inhibition of 26S proteasome beta 5 using LLVY as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307485((S)-2-azido-N-((S)-3-(3,5-bis(trifluoromethyl)phen...)
Affinity DataIC50: 130nMAssay Description:Inhibition of 26S proteasome beta 5 using LLVY as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307480(Pyrazine-2-carboxylic acid(1-[3-methyl-1-(2,9,9-tr...)
Affinity DataIC50: 160nMAssay Description:Inhibition of 26S proteasome beta 1 using nLPnLD as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307484((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50: 200nMAssay Description:Inhibition of 26S proteasome beta 5 using LLVY as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307486(5,5-difluoro-1,3,7,9-tetramethyl-10-(4-(1-((S)-1-(...)
Affinity DataIC50: 300nMAssay Description:Inhibition of 26S proteasome beta 5 using LLVY as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307479(Pyrazine-2-carboxylic acid(1-[3-methyl-1-(2,9,9-tr...)
Affinity DataIC50: 440nMAssay Description:Inhibition of 26S proteasome beta 1 using nLPnLD as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of 26S proteasome beta 2 using RLR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307486(5,5-difluoro-1,3,7,9-tetramethyl-10-(4-(1-((S)-1-(...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 26S proteasome beta 1 using nLPnLD as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307486(5,5-difluoro-1,3,7,9-tetramethyl-10-(4-(1-((S)-1-(...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 26S proteasome beta 2 using RLR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307480(Pyrazine-2-carboxylic acid(1-[3-methyl-1-(2,9,9-tr...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of 26S proteasome beta 2 using RLR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307485((S)-2-azido-N-((S)-3-(3,5-bis(trifluoromethyl)phen...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of 26S proteasome beta 2 using RLR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307485((S)-2-azido-N-((S)-3-(3,5-bis(trifluoromethyl)phen...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of 26S proteasome beta 1 using nLPnLD as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307483((S)-2-azido-N-((S)-1-((S)-3-(3,5-bis(trifluorometh...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of 26S proteasome beta 1 using nLPnLD as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307484((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of 26S proteasome beta 2 using RLR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307484((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of 26S proteasome beta 1 using nLPnLD as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307483((S)-2-azido-N-((S)-1-((S)-3-(3,5-bis(trifluorometh...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of 26S proteasome beta 2 using RLR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307482((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of 26S proteasome beta 2 using RLR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307482((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of 26S proteasome beta 1 using nLPnLD as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of 26S proteasome beta 1 using nLPnLD as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307479(Pyrazine-2-carboxylic acid(1-[3-methyl-1-(2,9,9-tr...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of 26S proteasome beta 2 using RLR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed