Compile Data Set for Download or QSAR
Report error Found 97 Enz. Inhib. hit(s) with all data for entry = 50005140
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488457(CHEMBL2286430)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488472(CHEMBL2286435)
Affinity DataEC50:  9.55E+3nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488445(CHEMBL2286440)
Affinity DataEC50:  2.04E+3nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488468(CHEMBL2286448)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488461(CHEBI:38451 | Halofenozide)
Affinity DataEC50:  78nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488460(CHEBI:38450 | Chromafenozide)
Affinity DataEC50:  1nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50178982(CHEMBL2228438)
Affinity DataEC50:  200nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488475(CHEMBL2286422)
Affinity DataEC50:  145nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488474(CHEMBL2286423)
Affinity DataEC50:  129nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488473(CHEMBL2286426)
Affinity DataEC50:  151nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488458(CHEMBL2286427)
Affinity DataEC50:  31nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488476(CHEMBL2286429)
Affinity DataEC50:  339nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488440(CHEMBL2228849)
Affinity DataEC50:  11nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488472(CHEMBL2286435)
Affinity DataEC50:  7.76E+3nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488454(CHEMBL2286436)
Affinity DataEC50:  2.88E+3nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488471(CHEMBL2286437)
Affinity DataEC50:  1.18E+3nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488452(CHEMBL2286442)
Affinity DataEC50:  1.78E+3nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488451(CHEMBL2286443)
Affinity DataEC50:  447nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488470(CHEMBL2286444)
Affinity DataEC50:  33nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488453(CHEMBL2286439)
Affinity DataEC50:  1.15E+3nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488469(CHEMBL2286410)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488449(CHEMBL2286446)
Affinity DataEC50:  427nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488475(CHEMBL2286422)
Affinity DataEC50:  288nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488459(CHEMBL2286421)
Affinity DataEC50:  3.63E+3nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488469(CHEMBL2286410)
Affinity DataEC50:  4.27E+3nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488466(CHEMBL2286418)
Affinity DataEC50:  5.50E+4nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50128305(N'-tert-butyl-N'-(3,5-dimethylbenzoyl)-3-methoxy-2...)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488456(CHEMBL2286431)
Affinity DataEC50:  17nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488448(CHEMBL2286411)
Affinity DataEC50:  3.55E+4nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488470(CHEMBL2286444)
Affinity DataEC50:  68nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488473(CHEMBL2286426)
Affinity DataEC50:  437nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488478(CHEMBL2286447)
Affinity DataEC50:  1.62E+4nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488478(CHEMBL2286447)
Affinity DataEC50:  7.76E+3nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50178990(CHEMBL2286425)
Affinity DataEC50:  309nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488467(CHEBI:38457 | RH-5849)
Affinity DataEC50:  437nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488446(CHEMBL2286424)
Affinity DataEC50:  324nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488476(CHEMBL2286429)
Affinity DataEC50:  135nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488455(CHEMBL2286434)
Affinity DataEC50:  1.91E+4nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488439(CHEMBL2286441)
Affinity DataEC50:  302nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488450(CHEMBL2286445)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50128314(N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-4-ethyl-be...)
Affinity DataEC50:  78nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488471(CHEMBL2286437)
Affinity DataEC50:  1.74E+3nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488443(CHEMBL2286420)
Affinity DataEC50:  794nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488474(CHEMBL2286423)
Affinity DataEC50:  437nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488446(CHEMBL2286424)
Affinity DataEC50:  457nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488455(CHEMBL2286434)
Affinity DataEC50:  2.19E+4nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488454(CHEMBL2286436)
Affinity DataEC50:  6.92E+3nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488442(CHEMBL2286438)
Affinity DataEC50:  339nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488453(CHEMBL2286439)
Affinity DataEC50:  1.12E+3nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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