Compile Data Set for Download or QSAR
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 50031242
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309658(N-(4-(5-cyano-7-(2-hydroxypropan-2-yl)benzo[d]oxaz...)
Affinity DataIC50: 28nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309627(N-(4-(5-cyanobenzo[d]oxazol-2-yl)phenyl)-2-(1,1,1,...)
Affinity DataIC50: 44nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309654(N-(4-(5-cyanobenzo[d]oxazol-2-yl)phenyl)-2-(1,1,1-...)
Affinity DataIC50: 51nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309653(N-(4-(5-cyanobenzo[d]oxazol-2-yl)phenyl)-2-(1,1,1,...)
Affinity DataIC50: 94nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50238385(N-(4-(5-cyanobenzo[d]oxazol-2-yl)phenyl)-2-(o-toly...)
Affinity DataIC50: 130nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309652(2-tert-butoxy-N-(4-(5-cyanobenzo[d]oxazol-2-yl)phe...)
Affinity DataIC50: 132nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309655(N-(4-(5-cyanobenzo[d]oxazol-2-yl)phenyl)-2-(1,1,1,...)
Affinity DataIC50: 151nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309628(2-(4-(2-(1,1,1,3,3,3-hexafluoro-2-methylpropan-2-y...)
Affinity DataIC50: 151nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309649(N-(4-(5-cyanobenzo[d]oxazol-2-yl)phenyl)-2-(2-(tri...)
Affinity DataIC50: 505nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309651(N-(4-(5-cyanobenzo[d]oxazol-2-yl)phenyl)-2-isoprop...)
Affinity DataIC50: 613nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309661(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(3-(tr...)
Affinity DataIC50: 810nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309657(2-(4-(2-isopropoxyethylamino)phenyl)benzo[d]oxazol...)
Affinity DataIC50: 890nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50238420(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(o-tol...)
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309648(N-(4-(5-cyanobenzo[d]oxazol-2-yl)phenyl)-2-(2-meth...)
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309623(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(3-chl...)
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309650(N-(4-(5-cyanobenzo[d]oxazol-2-yl)phenyl)-2-ethoxya...)
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309639(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(4-(tr...)
Affinity DataIC50: 1.77E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309664(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(4-flu...)
Affinity DataIC50: 1.77E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309625(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(3-flu...)
Affinity DataIC50: 1.99E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309633(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(2-chl...)
Affinity DataIC50: 2.15E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309666(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(4-nit...)
Affinity DataIC50: 2.21E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309630(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(2-eth...)
Affinity DataIC50: 2.59E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309631(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(2-pro...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309629(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-phenox...)
Affinity DataIC50: 4.23E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309637(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(2-nit...)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309665(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(4-met...)
Affinity DataIC50: 4.57E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309632(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(2-(tr...)
Affinity DataIC50: 6.39E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309668(2-(benzyloxy)-N-(4-(5-chlorobenzo[d]oxazol-2-yl)ph...)
Affinity DataIC50: 6.54E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309662(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(4-chl...)
Affinity DataIC50: 6.81E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309667(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(pheny...)
Affinity DataIC50: 8.13E+3nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309626(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(3-met...)
Affinity DataIC50: 1.29E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309669(2-(benzylamino)-N-(4-(5-chlorobenzo[d]oxazol-2-yl)...)
Affinity DataIC50: 1.81E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309638(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(m-tol...)
Affinity DataIC50: 1.93E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309659(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(3-nit...)
Affinity DataIC50: 2.65E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309660(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(p-tol...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309663(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(4-cya...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309647(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-phenox...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309646(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-N-methyl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309645(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-1-phenyl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309644(4-(5-chlorobenzo[d]oxazol-2-yl)-N-(2-methylbenzyl)...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309643(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(pheny...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309642(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-3-phenyl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309641(1-benzyl-3-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309640(benzyl 4-(5-chlorobenzo[d]oxazol-2-yl)phenylcarbam...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309636(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(2-met...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309635(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(2-flu...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309634(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(2-cya...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309624(N-(4-(5-chlorobenzo[d]oxazol-2-yl)phenyl)-2-(3-cya...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50309656(4-(benzo[d]oxazol-2-yl)-N-(2-phenoxyethyl)aniline ...)
Affinity DataIC50: 7.59E+4nMAssay Description:Inhibition of CETP assessed as cholesteryl ester transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed