Compile Data Set for Download or QSAR
Report error Found 71 Enz. Inhib. hit(s) with all data for entry = 50031219
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309158((2R,3R)-N-((4-benzylthiazol-2-yl)methyl)-2,3-dihyd...)
Affinity DataKi:  8nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309147((2R,3R)-4-(2-(3-chlorophenyl)pyrrolidin-1-yl)-2,3-...)
Affinity DataKi:  11nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309161((2R,3R)-N-((4-((6-chlorocyclohexa-2,4-dienyl)methy...)
Affinity DataKi:  13nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309149((2R,3R)-2,3-dihydroxy-N-methyl-4-oxo-N-(2-(thiophe...)
Affinity DataKi:  13nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309167((2R,3R)-2,3-dihydroxy-4-oxo-4-((R)-2-phenylpyrroli...)
Affinity DataKi:  20nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309160((2R,3R)-N-((4-benzyloxazol-2-yl)methyl)-2,3-dihydr...)
Affinity DataKi:  22nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 10(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309147((2R,3R)-4-(2-(3-chlorophenyl)pyrrolidin-1-yl)-2,3-...)
Affinity DataKi:  29nMAssay Description:Inhibition of ADAM10More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309150((2R,3R)-2,3-dihydroxy-4-(2-(3-methoxyphenyl)pyrrol...)
Affinity DataKi:  33nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309151((2R,3R)-4-(2-(3-(dimethylamino)phenyl)pyrrolidin-1...)
Affinity DataKi:  41nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309157((2R,3R)-N-(2-(4-benzylthiazol-2-yl)ethyl)-2,3-dihy...)
Affinity DataKi:  48nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309171((2R,3R)-2,3-dihydroxy-4-(isoindolin-2-yl)-4-oxo-N-...)
Affinity DataKi:  66nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309154((2R,3R)-N-(2-(4-benzylthiophen-2-yl)ethyl)-2,3-dih...)
Affinity DataKi:  66nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309156((2R,3R)-N-(4-benzylbenzyl)-4-(2-(3-chlorophenyl)py...)
Affinity DataKi:  70nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309170((2R,3R)-4-(3,4-dihydroisoquinolin-2(1H)-yl)-2,3-di...)
Affinity DataKi:  91nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309155((2R,3R)-N-((4-benzylthiophen-2-yl)methyl)-4-(2-(4-...)
Affinity DataKi:  93nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309166((2R,3R)-2,3-dihydroxy-4-oxo-4-(2-phenylpyrrolidin-...)
Affinity DataKi:  96nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309153((2R,3R)-N-(benzofuran-2-ylmethyl)-2,3-dihydroxy-4-...)
Affinity DataKi:  140nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309153((2R,3R)-N-(benzofuran-2-ylmethyl)-2,3-dihydroxy-4-...)
Affinity DataKi:  160nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309145((2R,3R)-2,3-dihydroxy-4-oxo-4-(2-(thiazol-2-yl)pyr...)
Affinity DataKi:  164nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309144((2R,3R)-2,3-dihydroxy-4-oxo-4-(2-(pyridin-2-yl)pyr...)
Affinity DataKi:  188nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309142((2R,3R)-2,3-dihydroxy-N1-methyl-N1-((R)-1-phenylet...)
Affinity DataKi:  238nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309153((2R,3R)-N-(benzofuran-2-ylmethyl)-2,3-dihydroxy-4-...)
Affinity DataKi:  300nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309146((2R,3R)-4-(2-(2-chlorophenyl)pyrrolidin-1-yl)-2,3-...)
Affinity DataKi:  323nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309143((2R,3R)-2,3-dihydroxy-4-oxo-4-(2-phenylpiperidin-1...)
Affinity DataKi:  325nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 10(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309132((2R,3R)-4-(4-(2-chlorophenyl)piperazin-1-yl)-2,3-d...)
Affinity DataKi:  400nMAssay Description:Inhibition of ADAM10More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309132((2R,3R)-4-(4-(2-chlorophenyl)piperazin-1-yl)-2,3-d...)
Affinity DataKi:  400nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309131((2R,3R)-2,3-dihydroxy-4-(4-(3-methoxyphenyl)pipera...)
Affinity DataKi:  400nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309169((2R,3R)-2,3-dihydroxy-4-oxo-4-(3-phenylpyrrolidin-...)
Affinity DataKi:  456nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309159((2R,3R)-N-(2-(4-benzyloxazol-2-yl)ethyl)-2,3-dihyd...)
Affinity DataKi:  461nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309141((2R,3R)-2,3-dihydroxy-N1-methyl-N1-((S)-1-phenylet...)
Affinity DataKi:  487nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309153((2R,3R)-N-(benzofuran-2-ylmethyl)-2,3-dihydroxy-4-...)
Affinity DataKi:  510nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309154((2R,3R)-N-(2-(4-benzylthiophen-2-yl)ethyl)-2,3-dih...)
Affinity DataKi:  700nMAssay Description:Inhibition of MMP12More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309168((2R,3R)-2,3-dihydroxy-4-oxo-4-((S)-2-phenylpyrroli...)
Affinity DataKi:  725nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 10(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309153((2R,3R)-N-(benzofuran-2-ylmethyl)-2,3-dihydroxy-4-...)
Affinity DataKi:  734nMAssay Description:Inhibition of ADAM10More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309148((2R,3R)-4-(2-(4-chlorophenyl)pyrrolidin-1-yl)-2,3-...)
Affinity DataKi:  755nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309137((2R,3R)-N1-benzyl-2,3-dihydroxy-N1-methyl-N4-(2-(t...)
Affinity DataKi:  764nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309140((2R,3R)-2,3-dihydroxy-N1-methyl-N1-(pyridin-3-ylme...)
Affinity DataKi:  943nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309139((2R,3R)-N1-(furan-2-ylmethyl)-2,3-dihydroxy-N1-met...)
Affinity DataKi:  1.02E+3nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309133((2R,3R)-4-(4-benzylpiperidin-1-yl)-2,3-dihydroxy-4...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309163((2R,3R)-N-((4-(2-chlorobenzyl)thiophen-2-yl)methyl...)
Affinity DataKi:  1.11E+3nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309138((2R,3R)-2,3-dihydroxy-N1-methyl-N1-phenethyl-N4-(2...)
Affinity DataKi:  1.28E+3nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309136((2R,3R)-2,3-dihydroxy-N1,N1-dimethyl-N4-(2-(thioph...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309134((2R,3R)-N1-cyclohexyl-2,3-dihydroxy-N1-methyl-N4-(...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309152((2R,3R)-N-benzyl-4-(2-(3-chlorophenyl)pyrrolidin-1...)
Affinity DataKi:  1.44E+3nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309162((2R,3R)-N-((4-(2-chlorobenzyl)thiophen-2-yl)methyl...)
Affinity DataKi:  1.52E+3nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309135((2R,3R)-2,3-dihydroxy-4-oxo-4-(4-(pyridin-2-yl)pip...)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309154((2R,3R)-N-(2-(4-benzylthiophen-2-yl)ethyl)-2,3-dih...)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309164((2R,3R)-2,3-dihydroxy-3-(thiazol-2-yl)-N-(2-(thiop...)
Affinity DataKi:  5.53E+3nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetMatrilysin(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309154((2R,3R)-N-(2-(4-benzylthiophen-2-yl)ethyl)-2,3-dih...)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of MMP7More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50309132((2R,3R)-4-(4-(2-chlorophenyl)piperazin-1-yl)-2,3-d...)
Affinity DataKi:  7.00E+3nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
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