Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50031205
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50300214(2-(4-(3,5-dichlorophenylcarbamothioyl)piperazin-1-...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of autotaxin-mediated pNP-TMP hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308960(2-(4-(9H-xanthene-9-carbonylcarbamothioyl)piperazi...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of autotaxin-mediated FS3 hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308961(4-(2-(3-ethyl-4-oxo-3,4,6,7,8,9-hexahydropyrimido[...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of autotaxin-mediated FS3 hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50300214(2-(4-(3,5-dichlorophenylcarbamothioyl)piperazin-1-...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of autotaxin-mediated FS3 hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308960(2-(4-(9H-xanthene-9-carbonylcarbamothioyl)piperazi...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of autotaxin-mediated pNP-TMP hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308958(4-(4-(2-(naphthalen-1-yl)-1,3-dioxoisoindoline-6-c...)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of autotaxin-mediated pNP-TMP hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308958(4-(4-(2-(naphthalen-1-yl)-1,3-dioxoisoindoline-6-c...)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of autotaxin-mediated FS3 hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308959(4,4'-(5,5'-carbonylbis(1,3-dioxoisoindoline-5,2-di...)
Affinity DataIC50: 1.28E+4nMAssay Description:Inhibition of autotaxin-mediated FS3 hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308957(3-{[1,3-dioxo-2-(4-phenylazo-phenyl)-2,3-dihydro-1...)
Affinity DataIC50: 1.28E+4nMAssay Description:Inhibition of autotaxin-mediated FS3 hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50300214(2-(4-(3,5-dichlorophenylcarbamothioyl)piperazin-1-...)
Affinity DataKi:  1.90E+3nMAssay Description:Competitive-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menten analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308960(2-(4-(9H-xanthene-9-carbonylcarbamothioyl)piperazi...)
Affinity DataKi:  2.70E+3nMAssay Description:Mixed-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menten analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308960(2-(4-(9H-xanthene-9-carbonylcarbamothioyl)piperazi...)
Affinity DataKi:  2.70E+3nMAssay Description:Competitive-type inhibition of autotaxin-mediated pNP-TMP hydrolysis by Michaelis-Menten analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308959(4,4'-(5,5'-carbonylbis(1,3-dioxoisoindoline-5,2-di...)
Affinity DataKi:  5.00E+3nMAssay Description:Competitive-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menten analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308958(4-(4-(2-(naphthalen-1-yl)-1,3-dioxoisoindoline-6-c...)
Affinity DataKi:  5.80E+3nMAssay Description:Mixed-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menten analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50300214(2-(4-(3,5-dichlorophenylcarbamothioyl)piperazin-1-...)
Affinity DataKi:  6.50E+3nMAssay Description:Noncompetitive inhibition of autotaxin-mediated pNP-TMP hydrolysis by Michaelis-Menten analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50300214(2-(4-(3,5-dichlorophenylcarbamothioyl)piperazin-1-...)
Affinity DataKi:  6.50E+3nMAssay Description:Noncompetitive inhibition of autotaxin-mediated pNP-TMP hydrolysis by Michaelis-Menten analysis for enzyme-substrate complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308961(4-(2-(3-ethyl-4-oxo-3,4,6,7,8,9-hexahydropyrimido[...)
Affinity DataKi:  6.50E+3nMAssay Description:Noncompetitive inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menten analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308961(4-(2-(3-ethyl-4-oxo-3,4,6,7,8,9-hexahydropyrimido[...)
Affinity DataKi:  9.30E+3nMAssay Description:Noncompetitive inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menten analysis for enzyme-substrate complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308957(3-{[1,3-dioxo-2-(4-phenylazo-phenyl)-2,3-dihydro-1...)
Affinity DataKi:  1.51E+4nMAssay Description:Mixed-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menten analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308960(2-(4-(9H-xanthene-9-carbonylcarbamothioyl)piperazi...)
Affinity DataKi:  1.98E+4nMAssay Description:Mixed-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menten analysis for enzyme-substrate complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308958(4-(4-(2-(naphthalen-1-yl)-1,3-dioxoisoindoline-6-c...)
Affinity DataKi:  3.23E+4nMAssay Description:Mixed-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menten analysis for enzyme-substrate complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Human)
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50308957(3-{[1,3-dioxo-2-(4-phenylazo-phenyl)-2,3-dihydro-1...)
Affinity DataKi:  4.03E+4nMAssay Description:Mixed-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menten analysis for enzyme-substrate complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed