Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50031199
LigandPNGBDBM50308835(4-((S)-2-(4-ethylthiazol-2-yl)-2-((S)-2-(methoxyca...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human protein-tyrosine phosphatase betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308854([7-(4-{1-Benzotriazol-1-yl-2-[4-(difluoro-phosphon...)
Affinity DataIC50: 5nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308841(Methanesulfonic acid 2-chloro-6-[3-hydroxy-4-(1,1,...)
Affinity DataIC50: 13nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308842(2-(4-Cyclohexylmethyl-2-fluoro-6-hydroxy-phenyl)-1...)
Affinity DataIC50: 14nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308847((S)-2-acetamido-3-(4-((3'-((isopropyl(4-(pentan-3-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308844(3-Fluoro-N-{1-{(R)-4-[2-(2-methanesulfonyl-phenoxy...)
Affinity DataIC50: 23nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM14269((S)-isothiazolidinone | N-[(1S)-1-(1H-1,3-benzodia...)
Affinity DataIC50: 25nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308844(3-Fluoro-N-{1-{(R)-4-[2-(2-methanesulfonyl-phenoxy...)
Affinity DataIC50: 25nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308845((S)-5-{4-[(S)-2-(1H-Benzoimidazol-2-yl)-2-(benzoth...)
Affinity DataIC50: 27nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50171117({4-[[3-Bromo-4-(difluoro-phosphono-methyl)-benzyl]...)
Affinity DataIC50: 28nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50171117({4-[[3-Bromo-4-(difluoro-phosphono-methyl)-benzyl]...)
Affinity DataIC50: 28nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50025835(CHEMBL592291)
Affinity DataIC50: 30nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM14269((S)-isothiazolidinone | N-[(1S)-1-(1H-1,3-benzodia...)
Affinity DataIC50: 32nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308854([7-(4-{1-Benzotriazol-1-yl-2-[4-(difluoro-phosphon...)
Affinity DataIC50: 36nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308835(4-((S)-2-(4-ethylthiazol-2-yl)-2-((S)-2-(methoxyca...)
Affinity DataIC50: 70nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308840(5-[2-Hydroxy-5-(1H-pyrrol-2-yl)-phenyl]-1,1-dioxo-...)
Affinity DataIC50: 80nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50142317((2-bromo-4-(3-oxo-2,3-diphenylpropyl)phenyl)difluo...)
Affinity DataIC50: 120nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50239833((3-bromo-7-cyanonaphthalen-2-yl)difluoromethylphos...)
Affinity DataIC50: 120nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50239833((3-bromo-7-cyanonaphthalen-2-yl)difluoromethylphos...)
Affinity DataIC50: 120nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50142317((2-bromo-4-(3-oxo-2,3-diphenylpropyl)phenyl)difluo...)
Affinity DataIC50: 120nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308839(5-[3'-(6-Fluoro-2,3-dihydro-indol-1-yl)-biphenyl-4...)
Affinity DataIC50: 130nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308846(N-{(S)-1-(1H-Benzoimidazol-2-yl)-2-[3-methyl-4-(1,...)
Affinity DataIC50: 140nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308846(N-{(S)-1-(1H-Benzoimidazol-2-yl)-2-[3-methyl-4-(1,...)
Affinity DataIC50: 150nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308845((S)-5-{4-[(S)-2-(1H-Benzoimidazol-2-yl)-2-(benzoth...)
Affinity DataIC50: 250nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308853(2,2'-(4,4'-(o-tolylsulfonylazanediyl)bis(methylene...)
Affinity DataIC50: 600nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50166434(1,2,5-THIADIAZOLIDIN-3-ONE-1,1-DIOXIDE | 1,1-Dioxo...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50166434(1,2,5-THIADIAZOLIDIN-3-ONE-1,1-DIOXIDE | 1,1-Dioxo...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50308838(N,N'-(4,4'-(1,4-phenylenebis(oxy))bis(4,1-phenylen...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50166435(5-(4-METHOXYBIPHENYL-3-YL)-1,2,5-THIADIAZOLIDIN-3-...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308848(2-(3-(2-(2-(4-chlorophenyl)-4-methylthiazol-5-yl)e...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308836(3-(3-Chloro-phenyl)-5-[1-(4-hydroxy-3-methoxy-5-ni...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM13461(N-[(3S)-3-(methylcarbamoyl)-2-{3-[3-(sulfoamino)ph...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308836(3-(3-Chloro-phenyl)-5-[1-(4-hydroxy-3-methoxy-5-ni...)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308837(Difluoro-[1,1',4',1'']terphenyl-3-yl-methanesulfon...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM13461(N-[(3S)-3-(methylcarbamoyl)-2-{3-[3-(sulfoamino)ph...)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308855((2R)-3-((2S)-1-(aminooxy)-3-(4-((((4-chlorobutyl)(...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM13996(4-amino-5-{3-[(1E)-3-[3-hydroxy-2-(methoxycarbonyl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50131550((S)-4-((S)-1-amino-3-(4-(difluoro(phosphono)methyl...)
Affinity DataKi:  2.40nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50219566(5-(3-(1-(benzylsulfonyl)piperidin-4-ylamino)phenyl...)
Affinity DataKi:  4nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50219566(5-(3-(1-(benzylsulfonyl)piperidin-4-ylamino)phenyl...)
Affinity DataKi:  5nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308852((S)-2-(N-(4-(2-acetamido-3-(4-(3-hydroxy-2-(methox...)
Affinity DataKi:  18nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308849((S)-2-(carboxyformamido)-7-((5-fluoro-1H-indole-2-...)
Affinity DataKi:  18nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50131550((S)-4-((S)-1-amino-3-(4-(difluoro(phosphono)methyl...)
Affinity DataKi:  26nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308852((S)-2-(N-(4-(2-acetamido-3-(4-(3-hydroxy-2-(methox...)
Affinity DataKi:  65nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308836(3-(3-Chloro-phenyl)-5-[1-(4-hydroxy-3-methoxy-5-ni...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of PTP1B by cell-based competitive inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM13996(4-amino-5-{3-[(1E)-3-[3-hydroxy-2-(methoxycarbonyl...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308843(5-{2-Methyl-5-[3-(1-phenylmethanesulfonyl-piperidi...)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308850(2-(4-((S)-2-(tert-butoxycarbonylamino)-3-(4-(3-hyd...)
Affinity DataKi:  8.40E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308851(2-{4-[2-ACETYLAMINO-3-(4-CARBOXYMETHOXY-3-HYDROXY-...)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
LigandPNGBDBM50308851(2-{4-[2-ACETYLAMINO-3-(4-CARBOXYMETHOXY-3-HYDROXY-...)
Affinity DataKi:  1.82E+5nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
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