Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50039032
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50366620(RESINIFERATOXIN)
Affinity DataEC50:  0.0190nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50305279([(1R,2R,6R,10S,11R,13S,15R,17R)-13-benzyl-6-hydrox...)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50305280([(1R,2R,6R,10S,11R,13S,15R,17R)-13-benzyl-6-hydrox...)
Affinity DataEC50:  17.4nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50305281([(1R,2R,6R,10S,11R,13S,15R,17R)-13-benzyl-6-hydrox...)
Affinity DataEC50:  0.650nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50305282([(1R,2R,6R,10S,11R,13S,15R,17R)-13-benzyl-6-hydrox...)
Affinity DataEC50:  0.980nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50305283([(1R,2R,6R,10S,11R,13S,15R,17R)-13-benzyl-6-hydrox...)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50305284([(1R,2R,6R,10S,11R,13S,15R,17R)-13-benzyl-6-hydrox...)
Affinity DataEC50:  13.7nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50305285([(1R,2R,6R,10S,11R,13S,15R,17R)-13-benzyl-6-hydrox...)
Affinity DataEC50:  0.00500nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM20461(Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50305278(iodoresiniferatoxin | CHEMBL595069)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed