Compile Data Set for Download or QSAR
Report error Found 57 Enz. Inhib. hit(s) with all data for entry = 50039002
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50241487(asiantic acid | 2,3,6,23-tetrahydroxyurs-12-en-28-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303478(N-[3-hydroxy-28-oxolup-20(29)-en-28-yl]glycine | [...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50240501((1R,3aS,5aR,5bR,7aR,9S,11aR,11bR,13aR)-methyl 9-hy...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303479(3alpha-isocyanato-1-isopropenyl-5alpha,5beta,8,8,1...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303480(N-cyclopropyl-N'-(9-hydroxy-1-isopropenyl-5alpha,5...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303481(N-(2-hydroxyethyl)-N'-(9-hydroxy-1-isopropenyl-5al...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303482(1-((1R,3alphaS,5alphaR,5betaR,9S,11alphaR)-icosahy...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303483(1-((1R,3alphaS,5alphaR,5betaR,9S,11alphaR)-icosahy...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303484(1-(2-(2-hydroxyethoxy)ethyl)-3-((1R,3alphaS,5alpha...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50241944(Lupenone | lupeone | CHEMBL486393)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50241943(Friedeline | friedelin | CHEMBL485998)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM23207((1R,2R,5S,8R,9R,10R,13R,14R,17S,19R)-5-(hydroxymet...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50218196(3-beta,28-Dihydroxy-urs-12-ene | urs-12-ene-3beta,...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50241956(urs-12-en-3beta-ol | alpha-amyrin | (3S,4aR,6aR,6b...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50250899(Arjunolic acid | (4aS,6aS,6bR,8aR,9R,10R,11R,12aR,...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303477(Ethyl N-[3-hydroxy-28-oxolup-20(29)-en-28-yl]glyci...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303447(Beta-glycyrrhetinic acid | CHEMBL579272)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303448(Beta-elemonic acid | CHEMBL566929)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50236238(5beta-cholanic acid-3alpha-ol | CHEMBL1478 | (3alp...)
Affinity DataEC50:  6.70E+3nMAssay Description:Agonist activity at human FXR expressed in COS1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50292431(Betulinic acid 3-O-succinate | 3-O-Succinyl-betuli...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303449(3-(Pent-4-enoyloxy)lup-20(29)-en-28-oic Acid | CHE...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303450(3-(Isobutyryloxy)lup-20(29)-en-28-oic Acid | CHEMB...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50240499((1R,3aS,5aR,5bR,11aR)-1-Isopropenyl-5a,5b,8,8,11a-...)
Affinity DataEC50:  4.71E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303451(1-Isopropenyl-5alpha,5beta,8,8,11alpha-pentamethyl...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303452(3-(Hydroxyimino)lup-20(29)-en-28-oic Acid | (1R,3a...)
Affinity DataEC50:  1.75E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303453(3-[(Acetyloxy)imino]lup-20(29)-en-28-oic Acid | CH...)
Affinity DataEC50:  5.00E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303454((5beta,8alpna,1beta,18beta,19beta)-3-[(Propionylox...)
Affinity DataEC50:  7.73E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303485((5beta,8alpha,14beta,18beta,19beta)-3-[(Benzoyloxy...)
Affinity DataEC50:  3.17E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303486((5beta,8apha,14beta,18beta,19beta)-3-[(Pent-4-enoy...)
Affinity DataEC50:  7.88E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303464(29-Dihydroxylupan-28-oic Acid | CHEMBL583203)
Affinity DataEC50:  3.32E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50236238(5beta-cholanic acid-3alpha-ol | CHEMBL1478 | (3alp...)
Affinity DataEC50:  5.60E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM23208(cid_64971 | CHEMBL269277 | (1R,2R,5S,8R,9R,10R,13R...)
Affinity DataEC50:  1.04E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50346601(Oleanolic acid (OA)(Compound 1) | NSC-114945 | OLE...)
Affinity DataEC50:  2.25E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50148911(3beta-hydroxyurs-12-en-28-oic acid | (3beta)-3-hyd...)
Affinity DataEC50:  1.43E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303455((5beta,8alpha,14beta,18beta,19beta)-3-[(Isobutyryl...)
Affinity DataEC50:  3.65E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303456(3-Methoxylupan-28-oic Acid | CHEMBL567770)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303457(Benzyl 3-Hydroxylup-20(29)-en-28-oate | CHEMBL5715...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303458(Benzyl 3-Methoxylup-20(29)-en-28-oate | CHEMBL5771...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303459((1R,3aS,5aR,5bR,7aR,9S,11aR,11bR,13aR,13bR)-9-ally...)
Affinity DataEC50:  2.08E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303460((1R,3aS,5aR,5bR,7aR,9R,11aR,11bR,13aR,13bR)-9-ally...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303461((1R,3aS,5aR,5bR,7aR,9S,11aR,11bR,13bR)-9-hydroxy-5...)
Affinity DataEC50:  6.27E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303462((1R,3aS,5aR,5bR,7aR,9R,11aR,11bR,13bR)-9-hydroxy-5...)
Affinity DataEC50:  420nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303463(9-Hydroxy-5alpha,5beta,8,8,11alpha-pentamethyl-1-(...)
Affinity DataEC50:  6.91E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50050950(Dihydrobetulinic acid | Betulinic acid | CHEMBL37)
Affinity DataEC50:  2.17E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50103962(1-Acetyl-9-hydroxy-5alpha,5beta,8,8,11alpha-pentam...)
Affinity DataEC50:  3.11E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303465(2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)ethyl 3-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303466(2-[(tert-butoxycarbonyl)amino]ethyl 3-hydroxylup-2...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303467(Pyridin-4-ylmethyl 3-hydroxylup-20(29)-en-28-oate ...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303468(({[3-hydroxy-28-oxolup-20(29)-en-28-yl]oxy}methyl)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303469(N-cyclopropyl-3-hydroxylup-20(29)-en-28-amide | CH...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
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