Compile Data Set for Download or QSAR
Report error Found 98 Enz. Inhib. hit(s) with all data for entry = 3466
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35129(5-vinyl-3-pyridinecarbonitrile, 14b)
Affinity DataIC50: 0.880nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35141(5-vinyl-3-pyridinecarbonitrile, 23)
Affinity DataIC50: 1.30nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35137(5-vinyl-3-pyridinecarbonitrile, 19)
Affinity DataIC50: 1.80nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35123(5-vinyl-3-pyridinecarbonitrile, 12b)
Affinity DataIC50: 2.20nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

LigandPNGBDBM35123(5-vinyl-3-pyridinecarbonitrile, 12b)
Affinity DataIC50: 2.5nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35127(5-vinyl-3-pyridinecarbonitrile, 13c)
Affinity DataIC50: 2.80nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

LigandPNGBDBM35155(5-vinyl-3-pyridinecarbonitrile, 37)
Affinity DataIC50: 3.40nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35140(5-vinyl-3-pyridinecarbonitrile, 22)
Affinity DataIC50: 3.5nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35154(5-vinyl-3-pyridinecarbonitrile, 36)
Affinity DataIC50: 3.60nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35128(5-vinyl-3-pyridinecarbonitrile, 14a)
Affinity DataIC50: 3.60nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35126(5-vinyl-3-pyridinecarbonitrile, 13b)
Affinity DataIC50: 4nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35135(5-vinyl-3-pyridinecarbonitrile, 17)
Affinity DataIC50: 4.90nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35130(5-vinyl-3-pyridinecarbonitrile, 14c)
Affinity DataIC50: 5.20nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35165(3-pyridinecarbonitrile, 48)
Affinity DataIC50: 5.20nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35136(5-vinyl-3-pyridinecarbonitrile, 18)
Affinity DataIC50: 5.70nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

LigandPNGBDBM35129(5-vinyl-3-pyridinecarbonitrile, 14b)
Affinity DataIC50: 5.80nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35132(5-vinyl-3-pyridinecarbonitrile, 15b)
Affinity DataIC50: 6nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35124(5-vinyl-3-pyridinecarbonitrile, 12c)
Affinity DataIC50: 6.40nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35138(5-vinyl-3-pyridinecarbonitrile, 20)
Affinity DataIC50: 6.80nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35151(5-vinyl-3-pyridinecarbonitrile, 33)
Affinity DataIC50: 7.40nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

LigandPNGBDBM35128(5-vinyl-3-pyridinecarbonitrile, 14a)
Affinity DataIC50: 8nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35139(5-vinyl-3-pyridinecarbonitrile, 21)
Affinity DataIC50: 8.90nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35134(5-vinyl-3-pyridinecarbonitrile, 16)
Affinity DataIC50: 9.30nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35125(5-vinyl-3-pyridinecarbonitrile, 13a)
Affinity DataIC50: 10nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35133(5-vinyl-3-pyridinecarbonitrile, 15c)
Affinity DataIC50: 11nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35160(5-vinyl-3-pyridinecarbonitrile, 42)
Affinity DataIC50: 11nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35158(5-vinyl-3-pyridinecarbonitrile, 40)
Affinity DataIC50: 12nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35159(5-vinyl-3-pyridinecarbonitrile, 41)
Affinity DataIC50: 12nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

LigandPNGBDBM35140(5-vinyl-3-pyridinecarbonitrile, 22)
Affinity DataIC50: 15nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

LigandPNGBDBM35126(5-vinyl-3-pyridinecarbonitrile, 13b)
Affinity DataIC50: 16nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35120(5-vinyl-3-pyridinecarbonitrile, 11b)
Affinity DataIC50: 16nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35142(5-vinyl-3-pyridinecarbonitrile, 24)
Affinity DataIC50: 16nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35164(5-vinyl-3-pyridinecarbonitrile, 47)
Affinity DataIC50: 17nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

LigandPNGBDBM35130(5-vinyl-3-pyridinecarbonitrile, 14c)
Affinity DataIC50: 18nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

LigandPNGBDBM35141(5-vinyl-3-pyridinecarbonitrile, 23)
Affinity DataIC50: 18nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35149(5-vinyl-3-pyridinecarbonitrile, 31)
Affinity DataIC50: 19nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35118(5-vinyl-3-pyridinecarbonitrile, 4c)
Affinity DataIC50: 19nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35143(5-vinyl-3-pyridinecarbonitrile, 25)
Affinity DataIC50: 22nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35144(5-vinyl-3-pyridinecarbonitrile, 26)
Affinity DataIC50: 22nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

LigandPNGBDBM35125(5-vinyl-3-pyridinecarbonitrile, 13a)
Affinity DataIC50: 22nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35145(5-vinyl-3-pyridinecarbonitrile, 27)
Affinity DataIC50: 23nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35150(5-vinyl-3-pyridinecarbonitrile, 32)
Affinity DataIC50: 24nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

LigandPNGBDBM35137(5-vinyl-3-pyridinecarbonitrile, 19)
Affinity DataIC50: 26nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

LigandPNGBDBM35127(5-vinyl-3-pyridinecarbonitrile, 13c)
Affinity DataIC50: 27nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

LigandPNGBDBM35134(5-vinyl-3-pyridinecarbonitrile, 16)
Affinity DataIC50: 28nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

LigandPNGBDBM35138(5-vinyl-3-pyridinecarbonitrile, 20)
Affinity DataIC50: 29nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35146(5-vinyl-3-pyridinecarbonitrile, 28)
Affinity DataIC50: 31nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35122(5-vinyl-3-pyridinecarbonitrile, 12a)
Affinity DataIC50: 31nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

LigandPNGBDBM35136(5-vinyl-3-pyridinecarbonitrile, 18)
Affinity DataIC50: 33nMAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

LigandPNGBDBM35121(5-vinyl-3-pyridinecarbonitrile, 11c)
Affinity DataIC50: 34nMpH: 7.2 T: 2°CAssay Description:All IC50s were measured by using a modified IMAP protocol from Molecular Devices. The kinase reaction was carried out in a Corning Costar 384 well pl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2009
Entry Details Article
PubMed
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