Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50030668
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414916(CHEMBL567005)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414917(CHEMBL567004)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414912(CHEMBL566532)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414918(CHEMBL567832)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414898(CHEMBL584268)
Affinity DataIC50: 14nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414914(CHEMBL577495)
Affinity DataIC50: 20nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414900(CHEMBL583636)
Affinity DataIC50: 28nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414901(CHEMBL567006)
Affinity DataIC50: 36nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414897(CHEMBL566767)
Affinity DataIC50: 47nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414904(CHEMBL565471)
Affinity DataIC50: 53nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM20842(3-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]-1,2-dihydroq...)
Affinity DataIC50: 54nMAssay Description:Inhibition of human CDK5More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414899(CHEMBL566114)
Affinity DataIC50: 55nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414903(CHEMBL583632)
Affinity DataIC50: 73nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM20819(3-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]-1,2,3,4-tetr...)
Affinity DataIC50: 79nMAssay Description:Inhibition of human CDK5More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414902(CHEMBL568084)
Affinity DataIC50: 112nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414915(CHEMBL566115)
Affinity DataIC50: 119nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50299869(ethyl 2-methyl-6-oxo-5-(2-(pyridin-4-yl)thiazol-4-...)
Affinity DataIC50: 131nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50299869(ethyl 2-methyl-6-oxo-5-(2-(pyridin-4-yl)thiazol-4-...)
Affinity DataIC50: 131nMAssay Description:Inhibition of human CDK5More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414905(CHEMBL565918)
Affinity DataIC50: 139nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414908(CHEMBL566994)
Affinity DataIC50: 157nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414913(CHEMBL578375)
Affinity DataIC50: 160nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414907(CHEMBL584506)
Affinity DataIC50: 198nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414910(CHEMBL567437)
Affinity DataIC50: 647nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414906(CHEMBL567223)
Affinity DataIC50: 672nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414909(CHEMBL568083)
Affinity DataIC50: 779nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50414911(CHEMBL565675)
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed