Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50030865
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303019(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50: 1.72nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303018(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50: 2.13nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303027(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50: 2.56nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303014(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50: 2.56nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303011(2-tert-butyl-5-(5-(4-chlorophenyl)-1-(2,4-dichloro...)
Affinity DataIC50: 2.83nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303022(2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(5-...)
Affinity DataIC50: 3.03nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303020(2-(5-(4-chlorophenyl)-3-(5-(1-(4-chlorophenyl)cycl...)
Affinity DataIC50: 3.23nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303017(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50: 3.69nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303028(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50: 3.70nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303009(2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(5-...)
Affinity DataIC50: 3.93nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303013(2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(5-...)
Affinity DataIC50: 4.14nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303029(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-3-(5-(...)
Affinity DataIC50: 4.21nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303025(2-(5-(4-bromophenyl)-3-(5-(1-(4-chlorophenyl)cyclo...)
Affinity DataIC50: 4.44nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303016(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-3-(5-(...)
Affinity DataIC50: 4.70nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303026(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-3-(5-(...)
Affinity DataIC50: 4.86nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303015(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50: 4.91nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303024(2-(5-(4-bromophenyl)-3-(5-tert-butyl-1,3,4-thiadia...)
Affinity DataIC50: 4.93nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303008(2-tert-butyl-5-(5-(4-chlorophenyl)-1-(2,4-dichloro...)
Affinity DataIC50: 6.47nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303023(2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-(5-...)
Affinity DataIC50: 7.39nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303012(2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(5-...)
Affinity DataIC50: 10.3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303010(2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-(5-...)
Affinity DataIC50: 14.7nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303021(2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-(5-...)
Affinity DataIC50: 26.9nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303019(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50: 38.5nMAssay Description:Binding affinity to human CB2 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataIC50: 92.5nMAssay Description:Binding affinity to human CB2 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303019(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50: 245nMAssay Description:Displacement of [3H]WIN-552122 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303014(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50: 414nMAssay Description:Displacement of [3H]WIN-552122 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303027(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50: 427nMAssay Description:Displacement of [3H]WIN-552122 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataIC50: 1.76E+3nMAssay Description:Displacement of [3H]WIN-552122 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303028(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]WIN-552122 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed