Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50004330
TargetProtease(Human immunodeficiency virus type 1)
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50371232(CARNOSIC ACID)
Affinity DataIC50: 240nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50232007(GANOMYCIN B)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of recombinant HIV1 protease after 30 mins by reverse phase HPLCMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50479301(CHEBI:66431 | Schisanlactone A)
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of HIV1 protease dimerization by Zhang-Poorman kinetic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50481851(Ganomycin I)
Affinity DataIC50: 2.19E+4nMAssay Description:Inhibition of recombinant HIV1 protease after 30 mins by reverse phase HPLCMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50067040(CHEMBL116438 | 1,7-bis(4-hydroxy-3-methoxyphenyl)1...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of HIV1 integrase 3' processing activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50067040(CHEMBL116438 | 1,7-bis(4-hydroxy-3-methoxyphenyl)1...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50067040(CHEMBL116438 | 1,7-bis(4-hydroxy-3-methoxyphenyl)1...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50232007(GANOMYCIN B)
Affinity DataKi:  4.00E+3nMAssay Description:Competitive inhibition of HIV1 protease by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50479301(CHEBI:66431 | Schisanlactone A)
Affinity DataKi:  1.75E+4nMAssay Description:Inhibition of HIV1 protease dimerization by Zhang-Poorman kinetic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed