Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50030852
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50036166(3-Pyridin-3-yl-1-aza-bicyclo[2.2.2]oct-2-ene | 3-(...)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]MLA from rat alpha7 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50036166(3-Pyridin-3-yl-1-aza-bicyclo[2.2.2]oct-2-ene | 3-(...)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]alpha-bungarotoxin from rat alpha7 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50302794(4-(5-(quinuclidin-3-yl)pyridin-2-yl)morpholine | C...)
Affinity DataKi:  350nMAssay Description:Displacement of [125I]alpha-bungarotoxin from rat alpha7 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50302796(4-(5-(1-azabicyclo[2.2.2]oct-2-en-3-yl)pyridin-2-y...)
Affinity DataKi:  400nMAssay Description:Displacement of [125I]alpha-bungarotoxin from rat alpha7 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50302795(1-methyl-3-(6-morpholinopyridin-3-yl)-1-azoniabicy...)
Affinity DataKi:  5.60E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from rat alpha7 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50302793(1-methyl-3-(6-morpholinopyridin-3-yl)-1-azoniabicy...)
Affinity DataKi:  6.10E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from rat alpha7 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50302797(4-(5-(7-azabicyclo[2.2.1]hept-2-en-2-yl)pyridin-2-...)
Affinity DataKi:  3.30E+4nMAssay Description:Displacement of [125I]alpha-bungarotoxin from rat alpha7 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed