Compile Data Set for Download or QSAR
Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 50039090
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50378699(CHEMBL1204023)
Affinity DataIC50: 80nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50158453(N-(3-Phenylamino-4-pyridinyl)trifluoromethanesulfo...)
Affinity DataIC50: 90nMAssay Description:Inhibition of COX2 in human whole bloodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50158453(N-(3-Phenylamino-4-pyridinyl)trifluoromethanesulfo...)
Affinity DataIC50: 90nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311366(N-[3-(4-methoxyphenylamino)-4-pyridinyl]trifluorom...)
Affinity DataIC50: 100nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311392(N-[3-(3-Bromophenylamino)-4-pyridinyl]trifluoromet...)
Affinity DataIC50: 120nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50120981(1,1,1-trifluoro-N-(3-phenoxypyridin-4-yl)methanesu...)
Affinity DataIC50: 140nMAssay Description:Inhibition of COX1 in human whole bloodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311366(N-[3-(4-methoxyphenylamino)-4-pyridinyl]trifluorom...)
Affinity DataIC50: 160nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311396(N-[3-(4-methylphenylamino)-4-pyridinyl]trifluorome...)
Affinity DataIC50: 170nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50158453(N-(3-Phenylamino-4-pyridinyl)trifluoromethanesulfo...)
Affinity DataIC50: 180nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50158453(N-(3-Phenylamino-4-pyridinyl)trifluoromethanesulfo...)
Affinity DataIC50: 180nMAssay Description:Inhibition of COX1 in human whole bloodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311389(N-[3-(2-chlorophenylamino)-4-pyridinyl]trifluorome...)
Affinity DataIC50: 190nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311398(N-[3-(3-ethylphenylamino)-4-pyridinyl]trifluoromet...)
Affinity DataIC50: 240nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311390(N-[3-(3-Chlorophenylamino)-4-pyridinyl]trifluorome...)
Affinity DataIC50: 270nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50378700(CHEMBL1204024)
Affinity DataIC50: 270nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50378699(CHEMBL1204023)
Affinity DataIC50: 330nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 350nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50120980(N-(3-phenoxypyridin-4-yl)methanesulfonamide | N-(3...)
Affinity DataIC50: 410nMAssay Description:Inhibition of COX1 in human whole bloodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311391(N-[3-(4-Chlorophenylamino)-4-pyridinyl]trifluorome...)
Affinity DataIC50: 410nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311395(N-[3-(3-Methylphenylamino)-4-pyridinyl]trifluorome...)
Affinity DataIC50: 450nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311396(N-[3-(4-methylphenylamino)-4-pyridinyl]trifluorome...)
Affinity DataIC50: 460nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311368(N-[3-(2-chlorophenylamino)-4-pyridinyl]methanesulf...)
Affinity DataIC50: 480nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311394(N-[3-(2-methylphenylamino)-4-pyridinyl]trifluorome...)
Affinity DataIC50: 480nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311373(N-[3-(2-methylphenylamino)-4-pyridinyl]methanesulf...)
Affinity DataIC50: 560nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311381(N-[3-(4-methoxyphenylamino)-4-pyridinyl]methanesul...)
Affinity DataIC50: 560nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50120981(1,1,1-trifluoro-N-(3-phenoxypyridin-4-yl)methanesu...)
Affinity DataIC50: 620nMAssay Description:Inhibition of COX2 in human whole bloodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311398(N-[3-(3-ethylphenylamino)-4-pyridinyl]trifluoromet...)
Affinity DataIC50: 690nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50056999(CHEMBL56367 | nimesulide)
Affinity DataIC50: 700nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311369(N-[3-(3-Chlorophenylamino)-4-pyridinyl]methanesulf...)
Affinity DataIC50: 730nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311386(N-(3-cycloheptylamino-4-pyridinyl)trifluoromethane...)
Affinity DataIC50: 760nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311393(N-[3-(4-bromophenylamino)-4-pyridinyl]trifluoromet...)
Affinity DataIC50: 910nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311392(N-[3-(3-Bromophenylamino)-4-pyridinyl]trifluoromet...)
Affinity DataIC50: 910nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311399(N-[3-(4-ethylphenylamino)-4-pyridinyl]trifluoromet...)
Affinity DataIC50: 910nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50378701(CHEMBL1204025)
Affinity DataIC50: 940nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311395(N-[3-(3-Methylphenylamino)-4-pyridinyl]trifluorome...)
Affinity DataIC50: 990nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311401(N-[3-(3-methoxyphenylamino)-4-pyridinyl]trifluorom...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311390(N-[3-(3-Chlorophenylamino)-4-pyridinyl]trifluorome...)
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311400(N-[3-(2-methoxyphenylamino)-4-pyridinyl]trifluorom...)
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311382(N-(3-cyclopentylamino-4-pyridinyl)trifluoromethane...)
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311391(N-[3-(4-Chlorophenylamino)-4-pyridinyl]trifluorome...)
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50158452(N-(3-(phenylthio)pyridin-4-yl)methanesulfonamide |...)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of COX2 in human whole bloodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311399(N-[3-(4-ethylphenylamino)-4-pyridinyl]trifluoromet...)
Affinity DataIC50: 1.22E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311375(N-[3-(4-methylphenylamino)-4-pyridinyl]methanesulf...)
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311370(N-[3-(4-chlorophenylamino)-4-pyridinyl]methanesulf...)
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311401(N-[3-(3-methoxyphenylamino)-4-pyridinyl]trifluorom...)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311393(N-[3-(4-bromophenylamino)-4-pyridinyl]trifluoromet...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311386(N-(3-cycloheptylamino-4-pyridinyl)trifluoromethane...)
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311388(N-(3-phenylamino-4-pyridinyl)3,3,3-trifluoropropan...)
Affinity DataIC50: 2.06E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311389(N-[3-(2-chlorophenylamino)-4-pyridinyl]trifluorome...)
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311372(N-[3-(4-bromophenylamino)-4-pyridinyl]methanesulfo...)
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Liege

Curated by ChEMBL
LigandPNGBDBM50311367(N-(3-phenylamino-4-pyridinyl)methanesulfonamide | ...)
Affinity DataIC50: 2.26E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
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