Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50030616
TargetAlpha-1B adrenergic receptor(Rat)
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataIC50: 0.190nMAssay Description:Displacement of [3H]prazosin from adrenergic Alpha-1B receptor in Wistar rat liver membrane after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataIC50: 0.254nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1A receptor in Wistar rat submaxillary gland after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50203564(CHEMBL537669 | Yohimbine Hydrochloride | cid_6169 ...)
Affinity DataIC50: 3.67nMAssay Description:Displacement of [3H]MK9112 from human recombinant adrenergic alpha2A receptor expressed in insect Sf9 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50203564(CHEMBL537669 | Yohimbine Hydrochloride | cid_6169 ...)
Affinity DataIC50: 27.1nMAssay Description:Displacement of radioligand from human adrenergic Alpha-2C receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50299208(4-amino-6-methyl-2-(3-(4-p-tolylpiperazin-1-yl)pro...)
Affinity DataIC50: 56nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1A receptor in Wistar rat submaxillary gland after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50299208(4-amino-6-methyl-2-(3-(4-p-tolylpiperazin-1-yl)pro...)
Affinity DataIC50: 102nMAssay Description:Displacement of [3H]prazosin from adrenergic Alpha-1B receptor in Wistar rat liver membrane after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50299208(4-amino-6-methyl-2-(3-(4-p-tolylpiperazin-1-yl)pro...)
Affinity DataIC50: 320nMAssay Description:Displacement of [3H]MK9112 from human recombinant adrenergic alpha2A receptor expressed in insect Sf9 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed