Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50030942
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304315(trans-3-Oxo-N-(2-phenyl-2H-1,2,3-triazol-4-yl)-3Hs...)
Affinity DataIC50: 0.890nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304301(trans-N-[1-(3-Fluorophenyl)-1H-pyrazol-3-yl]-3-oxo...)
Affinity DataIC50: 0.920nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304313(trans-3-Oxo-N-(2-phenyl-1,3-thiazol-4-yl)-3H-spiro...)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304298(trans-3-Oxo-N-(1-phenyl-1H-pyrazol-4-yl)-3H-spiro[...)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304300(trans-N-[1-(2-fluorophenyl)-3-pyrazolyl]-3-oxospir...)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304303(trans-3-Oxo-N-(5-phenylpyrazin-2-yl)-3H-spiro[2-be...)
Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Rat)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304297(trans-3-Oxo-N-(1-phenyl-1H-pyrazol-3-yl)-3H-spiro[...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of rat Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301656(trans-3-Oxo-N-(5-phenylpyrimidin-2-yl)-3H-spiro[6-...)
Affinity DataIC50: 1.80nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304316(trans-N-[1-(4-Fluorophenyl)-1H-pyrazol-3-yl]-3-oxo...)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301651(trans-3-Oxo-N-(5-phenylpyrimidin-2-yl)-3H-spiro[5-...)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301644(trans-3-Oxo-N-(5-phenylpyrimidin-2-yl)-3H-spiro[4-...)
Affinity DataIC50: 2.10nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304312(trans-3-Oxo-N-(5-phenylpyridin-2-yl)-3H-spiro[6-az...)
Affinity DataIC50: 2.10nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304310(trans-3-Oxo-N-(5-phenylisoxazol-3-yl)-3H-spiro[6-a...)
Affinity DataIC50: 2.10nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Rat)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304300(trans-N-[1-(2-fluorophenyl)-3-pyrazolyl]-3-oxospir...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of rat Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Rat)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304301(trans-N-[1-(3-Fluorophenyl)-1H-pyrazol-3-yl]-3-oxo...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of rat Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304309(trans-3-Oxo-N-(5-phenylpyrazin-2-yl)-3H-spiro[6-az...)
Affinity DataIC50: 2.20nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304314(trans-3-Oxo-N-(1-phenyl-1H-pyrazol-4-yl)-3H-spiro[...)
Affinity DataIC50: 2.20nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Rat)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304299(trans-3-Oxo-N-(1-phenyl-1H-pyrazol-3-yl)-3H-spiro[...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of rat Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304299(trans-3-Oxo-N-(1-phenyl-1H-pyrazol-3-yl)-3H-spiro[...)
Affinity DataIC50: 2.30nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304307(trans-3-Oxo-N-(5-phenylpyrazin-2-yl)-3H-spiro[5-az...)
Affinity DataIC50: 2.40nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304318(trans-3-Oxo-N-(5-phenylisoxazol-3-yl)-3H-spiro[7-a...)
Affinity DataIC50: 2.40nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Rat)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304302(3'-oxo-N-(5-phenylpyrazin-2-yl)-3'H-spiro[cyclohex...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of rat Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304311(trans-3-Oxo-N-(3-phenyl-1H-pyrazol-5-yl)-3H-spiro[...)
Affinity DataIC50: 2.70nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304305(trans-3-Oxo-N-(5-phenylisoxazol-3-yl)-3H-spiro[4-a...)
Affinity DataIC50: 2.80nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301641(trans-3-Oxo-N-(5-phenylpyrimidin-2-yl)-3H-spiro[7-...)
Affinity DataIC50: 2.90nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304308(trans-3-Oxo-N-(3-phenyl-1H-pyrazol-5-yl)-3H-spiro[...)
Affinity DataIC50: 2.90nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304317(trans-3-Oxo-N-(5-phenylpyrazin-2-yl)-3H-spiro[7-az...)
Affinity DataIC50: 3.90nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304304(trans-3-Oxo-N-(5-phenylpyrazin-2-yl)-3H-spiro[4-az...)
Affinity DataIC50: 4.20nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304297(trans-3-Oxo-N-(1-phenyl-1H-pyrazol-3-yl)-3H-spiro[...)
Affinity DataIC50: 4.40nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Rat)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304298(trans-3-Oxo-N-(1-phenyl-1H-pyrazol-4-yl)-3H-spiro[...)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of rat Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304306(trans-3-Oxo-N-(3-phenyl-1H-pyrazol-5-yl)-3H-spiro[...)
Affinity DataIC50: 5.40nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304319(trans-3-Oxo-N-(3-phenyl-1H-pyrazol-5-yl)-3H-spiro[...)
Affinity DataIC50: 26nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed