Compile Data Set for Download or QSAR
Report error Found 115 Enz. Inhib. hit(s) with all data for entry = 50048852
LigandPNGBDBM50030815(CHEMBL404594)
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50030815(CHEMBL404594)
Affinity DataIC50: 0.350nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228195(CHEBI:2719 | Angiotensin Ii)
Affinity DataIC50: 1.30nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228894(CHEMBL312754)
Affinity DataIC50: 1.60nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228195(CHEBI:2719 | Angiotensin Ii)
Affinity DataIC50: 4nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228894(CHEMBL312754)
Affinity DataIC50: 5.10nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50282396(PD-123319 | (S)-1-(4-Dimethylamino-3-methyl-benzyl...)
Affinity DataIC50: 34nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228885(CHEMBL109832)
Affinity DataIC50: 44nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228993(CHEMBL110804)
Affinity DataIC50: 50nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228974(CHEMBL111287)
Affinity DataIC50: 51nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50229004(CHEMBL326663)
Affinity DataIC50: 56nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50010361(CHEMBL292277 | PD 123177 | PD-123177 | (S)-1-(4-Am...)
Affinity DataIC50: 66nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50229014(CHEMBL110531)
Affinity DataIC50: 67nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50010359(CHEMBL294558 | PD-121981 | 5-diphenylcarbamoyl-1-(...)
Affinity DataIC50: 70nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50229001(CHEMBL114126)
Affinity DataIC50: 71nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228879(CHEMBL114347)
Affinity DataIC50: 85nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50229020(CHEMBL109678)
Affinity DataIC50: 85nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228998(CHEMBL321664)
Affinity DataIC50: 89nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228961(CHEMBL2112328)
Affinity DataIC50: 97nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228966(CHEMBL321667)
Affinity DataIC50: 98nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228931(CHEMBL321221)
Affinity DataIC50: 110nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50229008(CHEMBL109562)
Affinity DataIC50: 110nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228990(CHEMBL111046)
Affinity DataIC50: 120nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50229009(CHEMBL111977)
Affinity DataIC50: 120nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228878(CHEMBL109921)
Affinity DataIC50: 130nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228900(CHEMBL320336)
Affinity DataIC50: 130nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228928(CHEMBL326246)
Affinity DataIC50: 140nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228968(CHEMBL322259)
Affinity DataIC50: 140nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228884(CHEMBL112874)
Affinity DataIC50: 150nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228964(CHEMBL111253)
Affinity DataIC50: 150nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228878(CHEMBL109921)
Affinity DataIC50: 170nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228969(CHEMBL112970)
Affinity DataIC50: 190nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228896(CHEMBL326042)
Affinity DataIC50: 200nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50282396(PD-123319 | (S)-1-(4-Dimethylamino-3-methyl-benzyl...)
Affinity DataIC50: 210nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228880(CHEMBL111382)
Affinity DataIC50: 240nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228988(CHEMBL109446)
Affinity DataIC50: 240nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50229011(CHEMBL111478)
Affinity DataIC50: 260nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228887(CHEMBL419210)
Affinity DataIC50: 270nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228891(CHEMBL432964)
Affinity DataIC50: 290nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228899(CHEMBL111782)
Affinity DataIC50: 290nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228980(CHEMBL110471)
Affinity DataIC50: 290nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50229016(CHEMBL109979)
Affinity DataIC50: 300nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228893(CHEMBL2112497)
Affinity DataIC50: 340nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228901(CHEMBL111519)
Affinity DataIC50: 350nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228978(CHEMBL325936)
Affinity DataIC50: 350nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228900(CHEMBL320336)
Affinity DataIC50: 370nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228883(CHEMBL432794)
Affinity DataIC50: 400nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228975(CHEMBL323598)
Affinity DataIC50: 450nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228963(CHEMBL321000)
Affinity DataIC50: 460nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandPNGBDBM50228927(CHEMBL325185)
Affinity DataIC50: 510nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
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