Compile Data Set for Download or QSAR
Report error Found 104 Enz. Inhib. hit(s) with all data for entry = 50030300
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293905((S)-4-amino-5-(4-(4-(2,4-dichloro-3-((2,4-dimethyl...)
Affinity DataIC50: 0.0500nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Jerini

Curated by ChEMBL
LigandPNGBDBM50074986(N-(2-((4-chloro-2-cyano-3-((2-methylquinolin-8-ylo...)
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H]bradykinin from guinea pig B2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293902(1-{4-methyl-3-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 0.540nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293906((S)-4-carbamimidoyl-N-(4-(1-(2,4-dichloro-3-((2,4-...)
Affinity DataIC50: 0.670nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293904(1-((4-methyl-3-((2-methyl-4-(4-methyl-1H-pyrazol-5...)
Affinity DataIC50: 1.10nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293903(1-((3-((4-(5-chlorothiazol-4-yl)-2-methylquinolin-...)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293899(1-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 1.40nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50067301(FK-3657 | (E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[...)
Affinity DataIC50: 1.40nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293901(cyclohexanecarboxylic acid{4-methyl-3-[2-methyl-4-...)
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293890(N-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 2.30nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293891(3-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 2.80nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293897(1-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 3.60nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293900(N-{4-methyl-3-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293899(1-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293897(1-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 5.10nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293900(N-{4-methyl-3-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 5.40nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293895(acetic acid 5-chloro-4-[2-methyl-4-(2-methyl-2H-py...)
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293888(2-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 6.5nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293891(3-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 6.60nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293886(2-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 7.5nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293890(N-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 7.80nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293892(dimethyl-carbamic acid 5-chloro-4-[2-methyl-4-(2-m...)
Affinity DataIC50: 8.30nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293904(1-((4-methyl-3-((2-methyl-4-(4-methyl-1H-pyrazol-5...)
Affinity DataIC50: 8.70nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293902(1-{4-methyl-3-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 8.80nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293901(cyclohexanecarboxylic acid{4-methyl-3-[2-methyl-4-...)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293903(1-((3-((4-(5-chlorothiazol-4-yl)-2-methylquinolin-...)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293892(dimethyl-carbamic acid 5-chloro-4-[2-methyl-4-(2-m...)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293894(N-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293896(N-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 14nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293885(8-((3-chloro-5-(1-methyl-1H-imidazol-2-ylthio)pyri...)
Affinity DataIC50: 18nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293880(8-(3,5-dichloro-pyridin-4-ylmethoxy)-2-methyl-4-(4...)
Affinity DataIC50: 20nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293886(2-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293894(N-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293884(8-[3-chloro-5-(thiazol-2-ylsulfanyl)-pyridin-4-ylm...)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293866(8-(3,5-dichloro-pyridin-4-ylmethoxy)-2-methyl-4-py...)
Affinity DataIC50: 32nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293893(3-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 33nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293889(3-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 36nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293887(2-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 37nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293885(8-((3-chloro-5-(1-methyl-1H-imidazol-2-ylthio)pyri...)
Affinity DataIC50: 43nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293868(8-(3,5-dichloro-pyridin-4-ylmethoxy)-2-methyl-4-(2...)
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293884(8-[3-chloro-5-(thiazol-2-ylsulfanyl)-pyridin-4-ylm...)
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293877(8-(3,5-dichloro-pyridin-4-ylmethoxy)-2-methyl-4-(5...)
Affinity DataIC50: 64nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293874(8-(3,5-dichloro-pyridin-4-ylmethoxy)-2-methyl-4-(4...)
Affinity DataIC50: 67nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293871(8-(3,5-dichloro-pyridin-4-ylmethoxy)-2-methyl-4-(2...)
Affinity DataIC50: 68nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293880(8-(3,5-dichloro-pyridin-4-ylmethoxy)-2-methyl-4-(4...)
Affinity DataIC50: 70nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293889(3-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 73nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293887(2-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 76nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293876(8-(3,5-dichloro-pyridin-4-ylmethoxy)-2-methyl-4-th...)
Affinity DataIC50: 80nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293864(8-(3,5-dichloro-pyridin-4-ylmethoxy)-2-methyl-4-(1...)
Affinity DataIC50: 90nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Jerini

Curated by ChEMBL
LigandPNGBDBM50293888(2-{5-chloro-4-[2-methyl-4-(2-methyl-2H-pyrazol-3-y...)
Affinity DataIC50: 91nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
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