Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 5631
TargetSerum paraoxonase/arylesterase 1(Human)
Ataturk University

LigandPNGBDBM92331(Lornoxicam)
Affinity DataKi:  9.00E+3nM ΔG°:  -28.8kJ/mole IC50: 1.36E+5nMpH: 10.5 T: 2°CAssay Description:The enzyme assay was based on the estimation of p-nitrophenol at 412nm. The molar extinction coefficient of p-nitrophenol was used to calculate enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2012
Entry Details Article
PubMed
TargetSerum paraoxonase/arylesterase 1(Human)
Ataturk University

LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataKi:  9.70E+4nM ΔG°:  -22.9kJ/mole IC50: 1.95E+5nMpH: 10.5 T: 2°CAssay Description:The enzyme assay was based on the estimation of p-nitrophenol at 412nm. The molar extinction coefficient of p-nitrophenol was used to calculate enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2012
Entry Details Article
PubMed
TargetSerum paraoxonase/arylesterase 1(Human)
Ataturk University

LigandPNGBDBM92332(Tenoxicam)
Affinity DataKi:  3.06E+5nM ΔG°:  -20.1kJ/mole IC50: 3.40E+5nMpH: 10.5 T: 2°CAssay Description:The enzyme assay was based on the estimation of p-nitrophenol at 412nm. The molar extinction coefficient of p-nitrophenol was used to calculate enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2012
Entry Details Article
PubMed
TargetSerum paraoxonase/arylesterase 1(Human)
Ataturk University

LigandPNGBDBM50174201(ARTHROTEC | GP 45840 | SOLARAZE | Sodium; [2-(2,6-...)
Affinity DataKi:  8.05E+5nM ΔG°:  -17.7kJ/mole IC50: 1.64E+6nMpH: 10.5 T: 2°CAssay Description:The enzyme assay was based on the estimation of p-nitrophenol at 412nm. The molar extinction coefficient of p-nitrophenol was used to calculate enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2012
Entry Details Article
PubMed
TargetSerum paraoxonase/arylesterase 1(Human)
Ataturk University

LigandPNGBDBM50022271(2-(3-benzoylphenyl)propanoic acid | 2-(3-Benzoylph...)
Affinity DataKi:  1.30E+7nM ΔG°:  -10.8kJ/mole IC50: 6.23E+6nMpH: 10.5 T: 2°CAssay Description:The enzyme assay was based on the estimation of p-nitrophenol at 412nm. The molar extinction coefficient of p-nitrophenol was used to calculate enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2012
Entry Details Article
PubMed
TargetSerum paraoxonase/arylesterase 1(Human)
Ataturk University

LigandPNGBDBM92333(Lincomycine)
Affinity DataKi:  1.11E+7nM ΔG°:  -11.2kJ/mole IC50: 1.30E+7nMpH: 10.5 T: 2°CAssay Description:The enzyme assay was based on the estimation of p-nitrophenol at 412nm. The molar extinction coefficient of p-nitrophenol was used to calculate enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2012
Entry Details Article
PubMed