Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50030414
TargetSialidase-2(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM4706(2,3-didehydro-2-deoxy-N-acetylneuraminic acid | (2...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of human NEU2 transiently transfected in HEK293T cells by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetSialidase-3(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM4706(2,3-didehydro-2-deoxy-N-acetylneuraminic acid | (2...)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of human NEU3 transiently transfected in HEK293T cells by fluorimetric high-performance liquid chromatographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetSialidase-4(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM4706(2,3-didehydro-2-deoxy-N-acetylneuraminic acid | (2...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of human NEU4 transiently transfected in HEK293T cells by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetSialidase-1(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM4706(2,3-didehydro-2-deoxy-N-acetylneuraminic acid | (2...)
Affinity DataIC50: 1.43E+5nMAssay Description:Inhibition of human NEU1 transiently transfected in HEK293T cells by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetSialidase-2(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50295841(4-Acetamido-5-(biphenyl-4-ylcarboxamido)-2-fluorob...)
Affinity DataIC50: 5.52E+5nMAssay Description:Inhibition of human NEU2 transiently transfected in HEK293 cells by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetSialidase-3(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50295839(4,5-Diacetamido-2-fluoro benzoic acid | CHEMBL5394...)
Affinity DataIC50: 2.00E+6nMAssay Description:Inhibition of human NEU3 transiently transfected in HEK293 cells by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetSialidase-2(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50295840(4-Acetamido-5-(2-naphthamido)-2-fluoro benzoic aci...)
Affinity DataIC50: 1.37E+6nMAssay Description:Inhibition of human NEU2 transiently transfected in HEK293 cells by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetSialidase-2(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50295839(4,5-Diacetamido-2-fluoro benzoic acid | CHEMBL5394...)
Affinity DataIC50: 1.20E+6nMAssay Description:Inhibition of human NEU2 transiently transfected in HEK293 cells by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetSialidase-2(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50295841(4-Acetamido-5-(biphenyl-4-ylcarboxamido)-2-fluorob...)
Affinity DataKi:  3.07E+5nMAssay Description:Inhibition of human NEU2 transiently transfected in HEK293 cells by Line-Weaver Burk plottingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed