Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50032044
TargetG-protein coupled estrogen receptor 1(Human)
University of New Mexico Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50303804(cid_3136844 | CHEMBL583543 | (3aS,4R,9bR)-4-(6-bro...)
Affinity DataIC50: 185nMAssay Description:Antagonist activity at GPR30 in human SKBr3 cells assessed as inhibition of calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Mouse)
University of New Mexico Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50303804(cid_3136844 | CHEMBL583543 | (3aS,4R,9bR)-4-(6-bro...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to ERbeta receptor in mouse COS7 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Mouse)
University of New Mexico Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50303803(cid_5322399 | cid_3136849 | CHEMBL569766 | 1-((3aS...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to ERalpha receptor in mouse COS7 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed