Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50030525
TargetMu-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50297503(17-(cyclopropylmethyl)-3,14-dihydroxy-6beta-(N,N-d...)
Affinity DataKi:  0.560nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50297505(l7-(cyclopropylmethyl)-3,l4-dihydroxy-6beta-(((4-m...)
Affinity DataKi:  0.790nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50297506(l7-(cyclopropylmethyl)-3,l4-dihydroxy-6beta-((meth...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKappa-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50297505(l7-(cyclopropylmethyl)-3,l4-dihydroxy-6beta-(((4-m...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50297504(17-(cyclopropylmethyl)-3,14-dihydroxy-6beta-(N,N-d...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50001709(CHEMBL558140 | CHEMBL140278 | 4-cyclopropylmethyl-...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50297505(l7-(cyclopropylmethyl)-3,l4-dihydroxy-6beta-(((4-m...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKappa-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50297506(l7-(cyclopropylmethyl)-3,l4-dihydroxy-6beta-((meth...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKappa-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50001709(CHEMBL558140 | CHEMBL140278 | 4-cyclopropylmethyl-...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKappa-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50297503(17-(cyclopropylmethyl)-3,14-dihydroxy-6beta-(N,N-d...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKappa-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50297504(17-(cyclopropylmethyl)-3,14-dihydroxy-6beta-(N,N-d...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50297503(17-(cyclopropylmethyl)-3,14-dihydroxy-6beta-(N,N-d...)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50297506(l7-(cyclopropylmethyl)-3,l4-dihydroxy-6beta-((meth...)
Affinity DataKi:  93nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50001709(CHEMBL558140 | CHEMBL140278 | 4-cyclopropylmethyl-...)
Affinity DataKi:  213nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50297504(17-(cyclopropylmethyl)-3,14-dihydroxy-6beta-(N,N-d...)
Affinity DataKi:  334nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed