Compile Data Set for Download or QSAR
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 50028552
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277555(Benzyl 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4...)
Affinity DataIC50: 17.8nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277951(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(2,2-d...)
Affinity DataIC50: 21.2nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277914(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(2-eth...)
Affinity DataIC50: 24.8nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277949(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataIC50: 26.9nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278049(5-(4-Chlorophenyl)-N-(cyclohexanecarbonyl)-1-(2,4-...)
Affinity DataIC50: 30.4nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278000(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataIC50: 32.7nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278002(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-hexano...)
Affinity DataIC50: 33.5nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277950(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(2-eth...)
Affinity DataIC50: 43.1nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278003(N-Butyryl-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl...)
Affinity DataIC50: 43.7nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277764(5-(4-Chlorophenyl)-N-((2-cyclohexylacetamido)methy...)
Affinity DataIC50: 46.5nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277724(5-(4-Chlorophenyl)-N-(cyclohexanecarboxamidomethyl...)
Affinity DataIC50: 49.2nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277952(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(3,3-d...)
Affinity DataIC50: 53.4nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278050(5-(4-Chlorophenyl)-N-(cyclopentanecarbonyl)-1-(2,4...)
Affinity DataIC50: 67.2nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277725(5-(4-Chlorophenyl)-N-(cycloheptanecarboxamidomethy...)
Affinity DataIC50: 75.6nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277592(tert-Butyl 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataIC50: 82.5nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277591(Butyl 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-...)
Affinity DataIC50: 99.7nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277726(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataIC50: 102nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278052(5-(4-Chlorophenyl)-N-(cyclopropanecarbonyl)-1-(2,4...)
Affinity DataIC50: 124nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278051(5-(4-Chlorophenyl)-N-(cyclobutanecarbonyl)-1-(2,4-...)
Affinity DataIC50: 127nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277763(5-(4-Chlorophenyl)-N-((2-cyclopentylacetamido)meth...)
Affinity DataIC50: 138nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277456(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(hexyl...)
Affinity DataIC50: 138nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277554(N-(Benzylcarbamoyl)-5-(4-chlorophenyl)-1-(2,4-dich...)
Affinity DataIC50: 146nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277723(5-(4-Chlorophenyl)-N-(cyclobutanecarboxamidomethyl...)
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278001(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-isobut...)
Affinity DataIC50: 161nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277684(5-(4-Chlorophenyl)-N-(cyclohexanecarbonyl)-1-(2,4-...)
Affinity DataIC50: 167nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277643(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N,4-dime...)
Affinity DataIC50: 220nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277644(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(2,2-d...)
Affinity DataIC50: 227nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277646(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N,4-dime...)
Affinity DataIC50: 247nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277485(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(isopr...)
Affinity DataIC50: 253nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277645(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(2-eth...)
Affinity DataIC50: 265nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277593(Neopentyl 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl...)
Affinity DataIC50: 363nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278004(N-Acetyl-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)...)
Affinity DataIC50: 383nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277457(5-(4-Chlorophenyl)-N-(cyclohexylcarbamoyl)-1-(2,4-...)
Affinity DataIC50: 390nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277458(5-(4-Chlorophenyl)-N-(cycloheptylcarbamoyl)-1-(2,4...)
Affinity DataIC50: 750nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277686(N-(Butyramidomethyl)-5-(4-chlorophenyl)-1-(2,4-dic...)
Affinity DataIC50: 905nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277687(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(isobu...)
Affinity DataIC50: 951nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277685(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataIC50: 1.18E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277875(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(4-flu...)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277874(5-(4-Chlorophenyl)-N-(3-chlorophenylsulfonyl)-1-(2...)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277841(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataIC50: 3.64E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277876(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(3-flu...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277877(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277842(5-(4-Chlorophenyl)-N-(4-chlorophenylsulfonyl)-1-(2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277911(N-(Benzylsulfonyl)-5-(4-chlorophenyl)-1-(2,4-dichl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277912(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(ethyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277913(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(isopr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277840(N-(Butylsulfonyl)-5-(4-chlorophenyl)-1-(2,4-dichlo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50277553(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from CB1R in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed