Compile Data Set for Download or QSAR
Report error Found 67 Enz. Inhib. hit(s) with all data for entry = 3116
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28274(4-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 2nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28269(3-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 2nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28239(2-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 2nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28285(N-[4-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazo...)
Affinity DataIC50: 3nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28258(2-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 4nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28276(4-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 4nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28278(4-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 4nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28279(2-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 4nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28281(2-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 4nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28283(4-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 4nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28292(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl...)
Affinity DataIC50: 4nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28284(N-[4-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazo...)
Affinity DataIC50: 4nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28275(4-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 6nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28257(2-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 6nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28287(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl...)
Affinity DataIC50: 6nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28260(4-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 7nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28254(2-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 8nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28273(N-[3-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazo...)
Affinity DataIC50: 8nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28267(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl...)
Affinity DataIC50: 8nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28288(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl...)
Affinity DataIC50: 9nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28270(3-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 10nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28253(1-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 11nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28286(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl...)
Affinity DataIC50: 11nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28266(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl...)
Affinity DataIC50: 11nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28263(2-[4-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazo...)
Affinity DataIC50: 12nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28291(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl...)
Affinity DataIC50: 12nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28250(1-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 12nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28282(2-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 12nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28252(3-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 13nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28251(1-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 13nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28289(4-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 15nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28271(5-(3-aminophenyl)-7-{5-[(4-fluorophenyl)methyl]-1,...)
Affinity DataIC50: 15nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28256(5-[(dimethylsulfamoyl)amino]-7-{5-[(4-fluorophenyl...)
Affinity DataIC50: 15nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28249(1-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 15nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28280(4-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 18nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28277(4-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 18nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28240(1-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 19nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28255(N-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 19nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28262(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl...)
Affinity DataIC50: 19nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28268(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl...)
Affinity DataIC50: 20nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28293(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl...)
Affinity DataIC50: 21nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28248(4-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 23nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28290(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl...)
Affinity DataIC50: 23nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28242(1-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 25nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28304(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl...)
Affinity DataIC50: 27nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28244(N-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 28nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28264(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl...)
Affinity DataIC50: 29nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28265(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl...)
Affinity DataIC50: 30nMAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28245(ethyl 0-[(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxad...)
Affinity DataIC50: 33nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
Gsk

LigandPNGBDBM28247(1-(7-{5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2...)
Affinity DataIC50: 38nMpH: 7.2 T: 2°CAssay Description:Purified recombinant integrase was first combined in a complex with biotinylated donor DNA- streptavidin-coated SPA beads. The complex was preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2009
Entry Details Article
PubMed
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