Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50030267
TargetRetinoic acid receptor RXR-alpha(Mouse)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50293410((E)-3-[5'-(Adamant-1-yl)-2-chloro-4'-hydroxy-2'-me...)
Affinity DataEC50:  576nMAssay Description:Transactivation of Gal4-LBD fused mouse RXRalpha (218 to 467) transfected in african green monkey CV1 cells assessed as luciferase activity at after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Mouse)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50293411(2-[5'-(Adamant-1-yl)-2-chloro-4'-[(2-methoxyethoxy...)
Affinity DataEC50:  1.14E+3nMAssay Description:Transactivation of Gal4-LBD fused mouse RXRalpha (218 to 467) transfected in african green monkey CV1 cells assessed as luciferase activity at after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Mouse)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50293412(6-[5-(Adamant-1-yl)-4-[(2-methoxyethoxy)methoxy]-2...)
Affinity DataEC50:  667nMAssay Description:Transactivation of Gal4-LBD fused mouse RXRalpha (218 to 467) transfected in african green monkey CV1 cells assessed as luciferase activity at after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Mouse)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50293413((E)-3-[5'-(Adamant-1-yl)-2-chloro-4'-[(2-methoxyet...)
Affinity DataEC50:  600nMAssay Description:Transactivation of Gal4-LBD fused mouse RXRalpha (218 to 467) transfected in african green monkey CV1 cells assessed as luciferase activity at after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Mouse)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM31892(CHEMBL705 | 9-cis retinoic acid | alitretinoin | P...)
Affinity DataEC50:  200nMAssay Description:Transactivation of Gal4-LBD fused mouse RXRalpha (218 to 467) transfected in african green monkey CV1 cells assessed as luciferase activity at after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor RXR-alpha(Mouse)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataEC50:  40nMAssay Description:Transactivation of Gal4-LBD fused mouse RXRalpha (218 to 467) transfected in african green monkey CV1 cells assessed as luciferase activity at after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)