Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 3150
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28736(2-[2-chloro-4-({2-[4-(trifluoromethyl)phenoxymethy...)
Affinity DataEC50:  46.7nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28748(2-[2-methyl-4-({2-propyl-2-[4-(trifluoromethyl)phe...)
Affinity DataEC50:  8.60nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28747(2-{2-methyl-4-[({1-[4-(trifluoromethyl)phenoxymeth...)
Affinity DataEC50:  23.3nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28746(2-[2-methyl-4-({3-methyl-2-[4-(trifluoromethyl)phe...)
Affinity DataEC50:  22.4nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28745(2-{2-methyl-4-[({2-[4-(trifluoromethyl)phenoxymeth...)
Affinity DataEC50:  45.6nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28744(2-[4-({2,2-difluoro-3-[4-(trifluoromethyl)phenoxy]...)
Affinity DataEC50:  147nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28743(2-(4-{[(2E)-3-cyano-2-[4-(trifluoromethyl)phenoxym...)
Affinity DataEC50:  35.4nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28742(2-(2-methyl-4-{[(2E)-3-phenyl-2-[4-(trifluoromethy...)
Affinity DataEC50:  45.5nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28741(2-[4-({3,3-difluoro-2-[4-(trifluoromethyl)phenoxym...)
Affinity DataEC50:  69.6nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28740(2-[2-methyl-4-({2-[4-(trifluoromethyl)phenoxymethy...)
Affinity DataEC50:  249nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28739(2-[3-chloro-4-({2-[4-(trifluoromethyl)phenoxymethy...)
Affinity DataEC50: >500nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28738(2-[2-methoxy-4-({2-[4-(trifluoromethyl)phenoxymeth...)
Affinity DataEC50: >1.00E+3nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28737(2-[2-(trifluoromethyl)-4-({2-[4-(trifluoromethyl)p...)
Affinity DataEC50: >1.00E+3nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28724(2-(2-methyl-4-{[2-(phenoxymethyl)prop-2-en-1-yl]su...)
Affinity DataEC50:  711nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28735(2-[2-methyl-4-({2-methylidene-4-[4-(trifluoromethy...)
Affinity DataEC50:  26.8nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28734(2-(2-methyl-4-{[2-({[4-(trifluoromethyl)phenyl]sul...)
Affinity DataEC50:  54.3nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28733(2-(2-methyl-4-{[2-({[4-(trifluoromethyl)phenyl]ami...)
Affinity DataEC50: >500nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28732(2-[2-methyl-4-({2-[4-(trifluoromethoxy)phenoxymeth...)
Affinity DataEC50:  28.4nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28731(2-(4-{[2-(2,4-dichlorophenoxymethyl)prop-2-en-1-yl...)
Affinity DataEC50:  138nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28730(2-[4-({2-[4-(dimethylamino)phenoxymethyl]prop-2-en...)
Affinity DataEC50:  238nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28729(2-(4-{[2-(4-methoxyphenoxymethyl)prop-2-en-1-yl]su...)
Affinity DataEC50:  216nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28728(2-[4-({2-[4-chloro-3-(trifluoromethyl)phenoxymethy...)
Affinity DataEC50: >500nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28727(2-[2-methyl-4-({2-[4-(trifluoromethyl)phenoxymethy...)
Affinity DataEC50:  17.1nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28726(2-(4-{[2-(3,4-dichlorophenoxymethyl)prop-2-en-1-yl...)
Affinity DataEC50:  49.8nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM28725(2-(4-{[2-(4-chlorophenoxymethyl)prop-2-en-1-yl]sul...)
Affinity DataEC50:  65.5nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed