Compile Data Set for Download or QSAR
Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 50041673
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412996(CHEMBL477432)
Affinity DataEC50:  145nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413002(CHEMBL475077)
Affinity DataEC50:  81nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412986(CHEMBL474474)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413010(BAM-3200 | CHEMBL506884)
Affinity DataEC50:  794nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412989(CHEMBL474473)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413001(CHEMBL474272)
Affinity DataEC50:  398nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413000(CHEMBL451657)
Affinity DataEC50:  288nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412999(CHEMBL449189)
Affinity DataEC50:  132nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412998(CHEMBL476619)
Affinity DataEC50:  4.17E+3nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412988(CHEMBL477008)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412997(CHEMBL477643)
Affinity DataEC50:  8.13E+3nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412987(CHEMBL475965)
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412995(CHEMBL477431)
Affinity DataEC50:  589nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412983(CHEMBL458001)
Affinity DataEC50:  8.32E+3nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412984(CHEMBL458002)
Affinity DataEC50:  4.07E+3nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412985(CHEMBL458220)
Affinity DataEC50:  126nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412990(CHEMBL456481)
Affinity DataEC50:  2.63E+4nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412991(CHEMBL514267)
Affinity DataEC50:  2.09E+4nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412992(CHEMBL457788)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412993(CHEMBL457789)
Affinity DataEC50:  1.10E+4nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412994(CHEMBL517029)
Affinity DataEC50:  2.69E+3nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413009(CHEMBL499944)
Affinity DataEC50:  3.24E+4nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413008(CHEMBL474470)
Affinity DataEC50:  2.14E+3nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413003(CHEMBL475282)
Affinity DataEC50:  123nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413004(CHEMBL448975)
Affinity DataEC50:  107nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413005(CHEMBL476627)
Affinity DataEC50:  295nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413007(CHEMBL500240)
Affinity DataEC50:  7.08E+3nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413006(CHEMBL450183)
Affinity DataEC50:  5.75E+3nMAssay Description:Agonist activity at human MrgX1 receptor expressed in HEK293 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412984(CHEMBL458002)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412984(CHEMBL458002)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412987(CHEMBL475965)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412988(CHEMBL477008)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412983(CHEMBL458001)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412984(CHEMBL458002)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]5HT from 5HT2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412985(CHEMBL458220)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412983(CHEMBL458001)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412988(CHEMBL477008)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]5HT from 5HT2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412985(CHEMBL458220)
Affinity DataKi:  98nMAssay Description:Displacement of [3H]5HT from 5HT2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412983(CHEMBL458001)
Affinity DataKi:  155nMAssay Description:Displacement of [3H]5HT from 5HT2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412985(CHEMBL458220)
Affinity DataKi:  302nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412983(CHEMBL458001)
Affinity DataKi:  417nMAssay Description:Displacement of [3H]5HT from 5HT1D receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412985(CHEMBL458220)
Affinity DataKi:  457nMAssay Description:Displacement of [3H]5HT from 5HT1D receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412983(CHEMBL458001)
Affinity DataKi:  490nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412983(CHEMBL458001)
Affinity DataKi:  525nMAssay Description:Displacement of [3H]5HT from 5HT1B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412984(CHEMBL458002)
Affinity DataKi:  562nMAssay Description:Displacement of [3H]prazosin from adrenergic Alpha-1B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412985(CHEMBL458220)
Affinity DataKi:  589nMAssay Description:Displacement of [3H]5HT from 5HT1B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412983(CHEMBL458001)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]prazosin from adrenergic Alpha-1B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412984(CHEMBL458002)
Affinity DataKi:  741nMAssay Description:Displacement of [3H]5HT from 5HT1D receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412984(CHEMBL458002)
Affinity DataKi:  776nMAssay Description:Displacement of [3H]5HT from 5HT1B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412984(CHEMBL458002)
Affinity DataKi:  776nMAssay Description:Displacement of [125I]iodosulpiride from dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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