Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50027886
TargetGlycogen synthase kinase-3 beta(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50265885(3-(2-Ethoxycarbonylmethyl-3,5-dioxo-[1,2,4]thiadia...)
Affinity DataIC50: 467nMAssay Description:Inhibition of GSK3-beta by Z'-LYTE kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50266190(ethyl 2-(3,5-dioxo-4-(2-oxo-2-(piperidin-1-yl)ethy...)
Affinity DataIC50: 539nMAssay Description:Inhibition of GSK3-beta by Z'-LYTE kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50265884(KRM-189 | 4-(2-chloroethyl)-2-phenyl-1,2,4-thiadia...)
Affinity DataIC50: 548nMAssay Description:Inhibition of GSK3-beta by Z'-LYTE kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50265886(4-(2-Ethoxycarbonylmethyl-3,5-dioxo-[1,2,4]thiadia...)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of GSK3-beta by Z'-LYTE kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50266189(KRM-195 | 4-(4-fluorobenzyl)-2-phenethyl-1,2,4-thi...)
Affinity DataIC50: 1.86E+3nMAssay Description:Inhibition of GSK3-beta by Z'-LYTE kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50266190(ethyl 2-(3,5-dioxo-4-(2-oxo-2-(piperidin-1-yl)ethy...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50265885(3-(2-Ethoxycarbonylmethyl-3,5-dioxo-[1,2,4]thiadia...)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50265884(KRM-189 | 4-(2-chloroethyl)-2-phenyl-1,2,4-thiadia...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM7782(CHEMBL26241 | 4-Benzyl-2-ethyl-1,2,4-thiadiazolidi...)
Affinity DataIC50: 7.15E+3nMAssay Description:Inhibition of GSK3-beta by Z'-LYTE kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM7782(CHEMBL26241 | 4-Benzyl-2-ethyl-1,2,4-thiadiazolidi...)
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50266189(KRM-195 | 4-(4-fluorobenzyl)-2-phenethyl-1,2,4-thi...)
Affinity DataIC50: 3.87E+4nMAssay Description:Inhibition of PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50265886(4-(2-Ethoxycarbonylmethyl-3,5-dioxo-[1,2,4]thiadia...)
Affinity DataIC50: 4.83E+4nMAssay Description:Inhibition of PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed