Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50027632
TargetFree fatty acid receptor 4(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50240347((Z,Z,Z)-9,12,15-octadecatrienoic acid | cis,cis,ci...)
Affinity DataEC50:  2.60E+3nMAssay Description:Agonist activity at human GPR120-G-alpha-16 fusion protein expressed in Flp-in HEK293 cells assessed as effect on intracellular calcium concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50275055(4-{4-[2-(Phenyl-2-pyridinylamino)ethoxy]phenyl}but...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human GPR120-G-alpha-16 fusion protein expressed in Flp-in HEK293 cells assessed as effect on intracellular calcium concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50275055(4-{4-[2-(Phenyl-2-pyridinylamino)ethoxy]phenyl}but...)
Affinity DataEC50:  1.90E+4nMAssay Description:Agonist activity at human GPR40 expressed in T-REx HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50275158(4-{4-[2-(phenyl-2-thiazolylamino)ethoxy]phenyl}but...)
Affinity DataEC50:  2.10E+4nMAssay Description:Agonist activity at human GPR40 expressed in T-REx HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50275158(4-{4-[2-(phenyl-2-thiazolylamino)ethoxy]phenyl}but...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human GPR120-G-alpha-16 fusion protein expressed in Flp-in HEK293 cells assessed as effect on intracellular calcium concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50240347((Z,Z,Z)-9,12,15-octadecatrienoic acid | cis,cis,ci...)
Affinity DataEC50:  5.20E+3nMAssay Description:Agonist activity at human GPR40 expressed in T-REx HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed