Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50027580
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245838((rel)-(8-(bis(2-chlorophenyl)methyl)-3-(pyridin-2-...)
Affinity DataEC50:  156nMAssay Description:Agonist activity at human cloned nociceptin receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246403((rel)-(8-(bis(2-chlorophenyl)methyl)-3-phenyl-8-az...)
Affinity DataEC50:  483nMAssay Description:Agonist activity at human cloned nociceptin receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245975((rel)-N-((3-(4-fluorobenzyl)-8-(bis(2-chlorophenyl...)
Affinity DataEC50:  129nMAssay Description:Agonist activity at human cloned nociceptin receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246450((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-phenyl-8...)
Affinity DataEC50:  269nMAssay Description:Agonist activity at human cloned nociceptin receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245974((rel)-(3-(4-fluorobenzyl)-8-(bis(2-chlorophenyl)me...)
Affinity DataEC50:  124nMAssay Description:Agonist activity at human cloned nociceptin receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245891((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(6-metho...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245836((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(pyridin...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246401((rel)-8-(bis(2-chlorophenyl)methyl)-3-phenyl-8-aza...)
Affinity DataKi:  6nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245837((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(pyridin...)
Affinity DataKi:  6nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245838((rel)-(8-(bis(2-chlorophenyl)methyl)-3-(pyridin-2-...)
Affinity DataKi:  7nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245977((rel)-(8-(bis(2-chlorophenyl)methyl)-3-(pyridin-2-...)
Affinity DataKi:  7nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246402((rel)-(8-(bis(2-chlorophenyl)methyl)-3-phenyl-8-az...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246400((rel)-(8-(bis(2-chlorophenyl)methyl)-3-(6-methoxyp...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246562((rel)-(3-benzyl-8-(bis(2-chlorophenyl)methyl)-8-az...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246563((rel)-N-((3-benzyl-8-(bis(2-chlorophenyl)methyl)-8...)
Affinity DataKi:  12nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245975((rel)-N-((3-(4-fluorobenzyl)-8-(bis(2-chlorophenyl...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246403((rel)-(8-(bis(2-chlorophenyl)methyl)-3-phenyl-8-az...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245842((rel)-(8-(bis(2-chlorophenyl)methyl)-3-(piperidin-...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245978((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(6-metho...)
Affinity DataKi:  20nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246450((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-phenyl-8...)
Affinity DataKi:  20nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246451((rel)-methyl (8-(bis(2-chlorophenyl)methyl)-3-phen...)
Affinity DataKi:  20nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245889((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(6-fluor...)
Affinity DataKi:  24nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246027((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(5-bromo...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245892((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(piperid...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245888((rel)-(8-(bis(2-chlorophenyl)methyl)-3-(6-fluoropy...)
Affinity DataKi:  29nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246501((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(4-fluor...)
Affinity DataKi:  31nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245974((rel)-(3-(4-fluorobenzyl)-8-(bis(2-chlorophenyl)me...)
Affinity DataKi:  34nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245841((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(pyridin...)
Affinity DataKi:  35nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245823((rel)-N-((3-benzyl-8-(bis(2-chlorophenyl)methyl)-8...)
Affinity DataKi:  39nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246560((rel)-8-(bis(2-chlorophenyl)methyl)-5'-fluoro-8-az...)
Affinity DataKi:  39nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246503((rel)-(1S,5S)-8-(bis(2-chlorophenyl)methyl)-8-azas...)
Affinity DataKi:  50nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245979((rel)-(8-(bis(2-chlorophenyl)methyl)-3-(3-methylpy...)
Affinity DataKi:  50nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245824((rel)-(3-benzyl-8-(bis(2-chlorophenyl)methyl)-8-az...)
Affinity DataKi:  55nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245976((rel)-3-(4-fluorobenzyl)-8-(bis(2-chlorophenyl)met...)
Affinity DataKi:  58nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246026((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(5-metho...)
Affinity DataKi:  62nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246500((rel)-1-((8-(bis(2-chlorophenyl)methyl)-3-phenyl-8...)
Affinity DataKi:  68nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246453((rel)-8-(bis(2-chlorophenyl)methyl)-3-phenyl-3-(py...)
Affinity DataKi:  70nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246561((rel)-8-(bis(2-chlorophenyl)methyl)-5'-methyl-8-az...)
Affinity DataKi:  74nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245840((rel)-(8-(bis(2-chlorophenyl)methyl)-3-(pyridin-3-...)
Affinity DataKi:  82nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246028((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(5-(pipe...)
Affinity DataKi:  99nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245890((rel)-(8-(bis(2-chlorophenyl)methyl)-3-(6-fluoropy...)
Affinity DataKi:  104nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245825((rel)-3-benzyl-8-(bis(2-chlorophenyl)methyl)-3-(py...)
Affinity DataKi:  116nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246502((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(4-metho...)
Affinity DataKi:  118nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246400((rel)-(8-(bis(2-chlorophenyl)methyl)-3-(6-methoxyp...)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]diprenorphine from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245980((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(3-methy...)
Affinity DataKi:  173nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246452((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-phenyl-8...)
Affinity DataKi:  210nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50246024((rel)-(8-(bis(2-chlorophenyl)methyl)-3-(3-(piperid...)
Affinity DataKi:  245nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245891((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(6-metho...)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]diprenorphine from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245876((rel)-1-((3-benzyl-8-(bis(2-chlorophenyl)methyl)-8...)
Affinity DataKi:  336nMAssay Description:Displacement of [125I][Tyr14]nociceptin FQ from human cloned nociceptin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50245836((rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(pyridin...)
Affinity DataKi:  374nMAssay Description:Displacement of [3H]diprenorphine from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 76 total ) | Next | Last >>
Jump to: