Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50000778
TargetAdenosine receptor A1(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50009709(CHEMBL310377 | 4-Amino-5-butyl-1-(3-chloro-phenyl)...)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibitory concentration against R[3H]-N6-PIA binding to adenosine A1 receptors in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50009707(CHEMBL95318 | 4-Amino-5-butyl-1-phenyl-1,5-dihydro...)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibitory concentration against R[3H]-N6-PIA binding to adenosine A1 receptors in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50009708(CHEMBL98939 | 4-Amino-1-(3-chloro-phenyl)-5-propyl...)
Affinity DataIC50: 1.46E+4nMAssay Description:Inhibitory concentration against R[3H]-N6-PIA binding to adenosine A1 receptors in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50009704(CHEMBL99656 | 4-Amino-1-(3-chloro-phenyl)-5-methyl...)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibitory concentration against R[3H]-N6-PIA binding to adenosine A1 receptors in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50009709(CHEMBL310377 | 4-Amino-5-butyl-1-(3-chloro-phenyl)...)
Affinity DataIC50: 1.92E+4nMAssay Description:Inhibitory concentration against R[3H]-N6-PIA binding to adenosine A2 receptors in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50009705(CHEMBL319304 | 4-Amino-1,5-diphenyl-1,5-dihydro-py...)
Affinity DataIC50: 1.98E+4nMAssay Description:Inhibitory concentration against R[3H]-N6-PIA binding to adenosine A1 receptors in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50009706(CHEMBL95590 | 4-Amino-5-ethyl-1-phenyl-1,5-dihydro...)
Affinity DataIC50: 2.01E+4nMAssay Description:Inhibitory concentration against R[3H]-N6-PIA binding to adenosine A1 receptors in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50009705(CHEMBL319304 | 4-Amino-1,5-diphenyl-1,5-dihydro-py...)
Affinity DataIC50: 2.35E+4nMAssay Description:Inhibitory concentration against R[3H]-N6-PIA binding to adenosine A2 receptors in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50009707(CHEMBL95318 | 4-Amino-5-butyl-1-phenyl-1,5-dihydro...)
Affinity DataIC50: 2.48E+4nMAssay Description:Inhibitory concentration against R[3H]-N6-PIA binding to adenosine A2 receptors in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50009708(CHEMBL98939 | 4-Amino-1-(3-chloro-phenyl)-5-propyl...)
Affinity DataIC50: 4.73E+4nMAssay Description:Inhibitory concentration against R[3H]-N6-PIA binding to adenosine A2 receptors in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50009710(CHEMBL95589 | 4-Amino-1-phenyl-5-propyl-1,5-dihydr...)
Affinity DataIC50: 5.02E+4nMAssay Description:Inhibitory concentration against R[3H]-N6-PIA binding to adenosine A2 receptors in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50009710(CHEMBL95589 | 4-Amino-1-phenyl-5-propyl-1,5-dihydr...)
Affinity DataIC50: 5.07E+4nMAssay Description:Inhibitory concentration against R[3H]-N6-PIA binding to adenosine A1 receptors in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50009706(CHEMBL95590 | 4-Amino-5-ethyl-1-phenyl-1,5-dihydro...)
Affinity DataIC50: 8.18E+4nMAssay Description:Inhibitory concentration against R[3H]-N6-PIA binding to adenosine A2 receptors in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed