Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 3566
LigandPNGBDBM36411(PIK294 | CID24905149 | 2-((4-amino-3-(3-hydroxyphe...)
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36408(CID24905153 | 1-cyclobutyl-3-(3,4-dimethoxyphenyl)...)
Affinity DataIC50: 4nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
University of California San Francisco

LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataIC50: 8nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36408(CID24905153 | 1-cyclobutyl-3-(3,4-dimethoxyphenyl)...)
Affinity DataIC50: 17nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36408(CID24905153 | 1-cyclobutyl-3-(3,4-dimethoxyphenyl)...)
Affinity DataIC50: 47nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of California San Francisco

LigandPNGBDBM36410(CID24905148 | 1-cyclopentyl-3-(H-imidazo[1,2-a]pyr...)
Affinity DataIC50: 53nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36408(CID24905153 | 1-cyclobutyl-3-(3,4-dimethoxyphenyl)...)
Affinity DataIC50: 72nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataIC50: 100nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36408(CID24905153 | 1-cyclobutyl-3-(3,4-dimethoxyphenyl)...)
Affinity DataIC50: 130nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36408(CID24905153 | 1-cyclobutyl-3-(3,4-dimethoxyphenyl)...)
Affinity DataIC50: 130nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36408(CID24905153 | 1-cyclobutyl-3-(3,4-dimethoxyphenyl)...)
Affinity DataIC50: 170nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36408(CID24905153 | 1-cyclobutyl-3-(3,4-dimethoxyphenyl)...)
Affinity DataIC50: 170nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36411(PIK294 | CID24905149 | 2-((4-amino-3-(3-hydroxyphe...)
Affinity DataIC50: 200nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36408(CID24905153 | 1-cyclobutyl-3-(3,4-dimethoxyphenyl)...)
Affinity DataIC50: 340nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataIC50: 410nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataIC50: 410nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36411(PIK294 | CID24905149 | 2-((4-amino-3-(3-hydroxyphe...)
Affinity DataIC50: 670nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR/Tyrosine-protein kinase HCK(Human)
University of California San Francisco

LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataIC50: 1.20E+3nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36410(CID24905148 | 1-cyclopentyl-3-(H-imidazo[1,2-a]pyr...)
Affinity DataIC50: 1.40E+3nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36408(CID24905153 | 1-cyclobutyl-3-(3,4-dimethoxyphenyl)...)
Affinity DataIC50: 1.40E+3nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataIC50: 1.40E+3nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataIC50: 1.50E+3nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36408(CID24905153 | 1-cyclobutyl-3-(3,4-dimethoxyphenyl)...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36408(CID24905153 | 1-cyclobutyl-3-(3,4-dimethoxyphenyl)...)
Affinity DataIC50: 2.30E+3nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36410(CID24905148 | 1-cyclopentyl-3-(H-imidazo[1,2-a]pyr...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36410(CID24905148 | 1-cyclopentyl-3-(H-imidazo[1,2-a]pyr...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36408(CID24905153 | 1-cyclobutyl-3-(3,4-dimethoxyphenyl)...)
Affinity DataIC50: 3.00E+3nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEphrin type-B receptor 4/Serine/threonine-protein kinase mTOR(Human)
University of California San Francisco

LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataIC50: 3.40E+3nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR/Tyrosine-protein kinase ABL1(Human)
University of California San Francisco

LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataIC50: 3.60E+3nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor protein-tyrosine kinase/Serine/threonine-protein kinase mTOR(Human)
University of California San Francisco

LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataIC50: 4.40E+3nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36410(CID24905148 | 1-cyclopentyl-3-(H-imidazo[1,2-a]pyr...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataIC50: 5.10E+3nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36410(CID24905148 | 1-cyclopentyl-3-(H-imidazo[1,2-a]pyr...)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36408(CID24905153 | 1-cyclobutyl-3-(3,4-dimethoxyphenyl)...)
Affinity DataIC50: 7.00E+3nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit/Tyrosine-protein kinase HCK(Human)
University of California San Francisco

LigandPNGBDBM36410(CID24905148 | 1-cyclopentyl-3-(H-imidazo[1,2-a]pyr...)
Affinity DataIC50: 8.90E+3nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36411(PIK294 | CID24905149 | 2-((4-amino-3-(3-hydroxyphe...)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36410(CID24905148 | 1-cyclopentyl-3-(H-imidazo[1,2-a]pyr...)
Affinity DataIC50: 1.10E+4nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36410(CID24905148 | 1-cyclopentyl-3-(H-imidazo[1,2-a]pyr...)
Affinity DataIC50: 1.20E+4nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit/Tyrosine-protein kinase ABL1(Human)
University of California San Francisco

LigandPNGBDBM36410(CID24905148 | 1-cyclopentyl-3-(H-imidazo[1,2-a]pyr...)
Affinity DataIC50: 1.30E+4nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36410(CID24905148 | 1-cyclopentyl-3-(H-imidazo[1,2-a]pyr...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36411(PIK294 | CID24905149 | 2-((4-amino-3-(3-hydroxyphe...)
Affinity DataIC50: 1.70E+4nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36411(PIK294 | CID24905149 | 2-((4-amino-3-(3-hydroxyphe...)
Affinity DataIC50: 1.70E+4nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit/Ephrin type-B receptor 4(Human)
University of California San Francisco

LigandPNGBDBM36410(CID24905148 | 1-cyclopentyl-3-(H-imidazo[1,2-a]pyr...)
Affinity DataIC50: 2.10E+4nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36411(PIK294 | CID24905149 | 2-((4-amino-3-(3-hydroxyphe...)
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36411(PIK294 | CID24905149 | 2-((4-amino-3-(3-hydroxyphe...)
Affinity DataIC50: 5.00E+4nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36411(PIK294 | CID24905149 | 2-((4-amino-3-(3-hydroxyphe...)
Affinity DataIC50: 5.00E+4nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36411(PIK294 | CID24905149 | 2-((4-amino-3-(3-hydroxyphe...)
Affinity DataIC50: 5.00E+4nMAssay Description:The assays were performed in 96-well microtiter plates that had been coated with a polyGluTyr peptide. Negative control wells received buffer alone w...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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