Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50027098
TargetHistamine H3 receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247055(1-(3-(3-phenylpropoxy)propyl)piperidine | CHEMBL46...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human histamine H3 receptor expressed in rat C6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247148(1-[3-(4-tert-Butylphenoxy)propyl]-4-piperidino-pip...)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247120(1-[2-(3-Methoxyphenoxy)ethyl]-4-piperidino-piperid...)
Affinity DataKi:  132nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247122(1-[2-(3-Trifluoromethylphenoxy)ethyl]-4-piperidino...)
Affinity DataKi:  164nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247125(1-[3-(4-Chlorophenoxy)propyl]-4-piperidino-piperid...)
Affinity DataKi:  165nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247124(1-[2-(4-Chlorophenoxy)ethyl]-4-piperidino-piperidi...)
Affinity DataKi:  176nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247093(1-[2-(3-Chlorophenoxy)ethyl]-4-piperidino-piperidi...)
Affinity DataKi:  235nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247089(4-Propyl-1-[3-(phenylpropoxy)propyl]piperidine | C...)
Affinity DataKi:  249nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247090(4-Butyl-1-[3-(phenylpropoxy)propyl]piperidine | CH...)
Affinity DataKi:  274nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247123(1-[2-(4-Methylphenoxy)ethyl]-4-piperidino-piperidi...)
Affinity DataKi:  300nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247091(4-Benzyl-1-[3-phenylpropoxy)propyl]piperidine | CH...)
Affinity DataKi:  326nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247092(2-[3-(3-phenylpropoxy)propyl]decahydroisoquinoline...)
Affinity DataKi:  393nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247088(2-[3-(3-Phenylpropoxy)propyl]-1,2,3,4-tetrahydro-i...)
Affinity DataKi:  560nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247121(1-[3-(3-Methoxyphenoxy)propyl]-4-piperidino-piperi...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed