Compile Data Set for Download or QSAR
Report error Found 71 Enz. Inhib. hit(s) with all data for entry = 50026669
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262214((2-((1H-indazol-6-yl)methylamino)phenyl)(5-methyl-...)
Affinity DataIC50: 52nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261960((2-((1H-indazol-6-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50: 74nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262274((2-((1H-indazol-6-yl)methylamino)phenyl)(6-methyl-...)
Affinity DataIC50: 76nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM21(VANDETANIB | N-(4-bromo-2-fluorophenyl)-6-methoxy-...)
Affinity DataIC50: 100nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261959((2-((1H-indazol-5-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50: 120nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261961((1H-indazol-3-yl)(2-(quinolin-6-ylmethylamino)phen...)
Affinity DataIC50: 130nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262057((2-((1H-indazol-6-yl)methylamino)phenyl)(1H-indol-...)
Affinity DataIC50: 140nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262105((5-methyl-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50: 160nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262057((2-((1H-indazol-6-yl)methylamino)phenyl)(1H-indol-...)
Affinity DataIC50: 170nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262106((1,5-dimethyl-1H-indol-3-yl)(2-(quinolin-6-ylmethy...)
Affinity DataIC50: 180nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261961((1H-indazol-3-yl)(2-(quinolin-6-ylmethylamino)phen...)
Affinity DataIC50: 230nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262056((2-((1H-indazol-5-yl)methylamino)phenyl)(1H-indol-...)
Affinity DataIC50: 240nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262054((2-((1H-indazol-6-yl)methylamino)phenyl)(1-methyl-...)
Affinity DataIC50: 250nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262277((2-((1H-indazol-6-yl)methylamino)phenyl)(5-fluoro-...)
Affinity DataIC50: 250nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262278((2-((1H-indazol-6-yl)methylamino)phenyl)(6-fluoro-...)
Affinity DataIC50: 250nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262274((2-((1H-indazol-6-yl)methylamino)phenyl)(6-methyl-...)
Affinity DataIC50: 250nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261960((2-((1H-indazol-6-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50: 270nMAssay Description:Inhibition of VEGFR1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262054((2-((1H-indazol-6-yl)methylamino)phenyl)(1-methyl-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261961((1H-indazol-3-yl)(2-(quinolin-6-ylmethylamino)phen...)
Affinity DataIC50: 300nMAssay Description:Inhibition of VEGFR1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262007((2-((1H-benzo[d]imidazol-5-yl)methylamino)phenyl)(...)
Affinity DataIC50: 310nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262275((2-((1H-indazol-6-yl)methylamino)phenyl)(7-methyl-...)
Affinity DataIC50: 355nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262157((5-methoxy-1H-indol-3-yl)(2-(quinolin-6-ylmethylam...)
Affinity DataIC50: 450nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261959((2-((1H-indazol-5-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50: 460nMAssay Description:Inhibition of VEGFR1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262106((1,5-dimethyl-1H-indol-3-yl)(2-(quinolin-6-ylmethy...)
Affinity DataIC50: 540nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262213((5-chloro-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50: 560nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262009((2-((1H-indazol-6-yl)methylamino)phenyl)(1-(2-meth...)
Affinity DataIC50: 560nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262056((2-((1H-indazol-5-yl)methylamino)phenyl)(1H-indol-...)
Affinity DataIC50: 610nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262158((6-methoxy-1H-indol-3-yl)(2-(quinolin-6-ylmethylam...)
Affinity DataIC50: 660nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262108((7-methyl-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50: 700nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262107((6-methyl-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50: 730nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261960((2-((1H-indazol-6-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50: 730nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261959((2-((1H-indazol-5-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50: 800nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262212((6-fluoro-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50: 810nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262331((2-((1H-indazol-6-yl)methylamino)phenyl)(5-chloro-...)
Affinity DataIC50: 830nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262214((2-((1H-indazol-6-yl)methylamino)phenyl)(5-methyl-...)
Affinity DataIC50: 870nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261904((1H-indazol-3-yl)(2-(pyridin-4-ylmethylamino)pheny...)
Affinity DataIC50: 870nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262107((6-methyl-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50: 940nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262275((2-((1H-indazol-6-yl)methylamino)phenyl)(7-methyl-...)
Affinity DataIC50: 950nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262058((1H-indol-3-yl)(2-(quinolin-6-ylmethylamino)phenyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262211((5-fluoro-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262331((2-((1H-indazol-6-yl)methylamino)phenyl)(5-chloro-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262278((2-((1H-indazol-6-yl)methylamino)phenyl)(6-fluoro-...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261904((1H-indazol-3-yl)(2-(pyridin-4-ylmethylamino)pheny...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262009((2-((1H-indazol-6-yl)methylamino)phenyl)(1-(2-meth...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262277((2-((1H-indazol-6-yl)methylamino)phenyl)(5-fluoro-...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261904((1H-indazol-3-yl)(2-(pyridin-4-ylmethylamino)pheny...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of VEGFR1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262212((6-fluoro-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262158((6-methoxy-1H-indol-3-yl)(2-(quinolin-6-ylmethylam...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262157((5-methoxy-1H-indol-3-yl)(2-(quinolin-6-ylmethylam...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262105((5-methyl-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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