Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50038638
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50262295(4-[(4R,7S,10S,13R)-10-(3-{[amino(iminiumyl)methyl]...)
Affinity DataEC50:  0.690nMAssay Description:Agonist activity at human NOP receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50106469(FGGFTCARKCARK | cyclo[Cys6,Cys10]N/OFQ(1-13)NH2 | ...)
Affinity DataEC50:  31nMAssay Description:Agonist activity at human NOP receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50106479(FGGFTGARKSARK | H-FGGFTGARKSARK-NH2 | NC(1-13)NH2 ...)
Affinity DataEC50:  0.780nMAssay Description:Agonist activity at human NOP receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50106479(FGGFTGARKSARK | H-FGGFTGARKSARK-NH2 | NC(1-13)NH2 ...)
Affinity DataEC50:  7.82nMAssay Description:Agonist activity at human NOP receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50262293([D-Asp7,Lys10]N/OFQ(1-13)NH2 | CHEMBL507653)
Affinity DataEC50:  106nMAssay Description:Agonist activity at human NOP receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50262292([Asp6,Lys10]N/OFQ(1-13)NH2 | CHEMBL507269)
Affinity DataEC50:  22.3nMAssay Description:Agonist activity at human NOP receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50262291(4-[(3S,6S,9S,17S)-6-(3-{[amino(iminiumyl)methyl]am...)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human NOP receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50262290(4-[(3S,6S,9S,12S,20S)-6-(3-{[amino(iminiumyl)methy...)
Affinity DataEC50:  4.12nMAssay Description:Agonist activity at human NOP receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50262295(4-[(4R,7S,10S,13R)-10-(3-{[amino(iminiumyl)methyl]...)
Affinity DataKi:  0.100nMAssay Description:Binding affinity to human NOP receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50262291(4-[(3S,6S,9S,17S)-6-(3-{[amino(iminiumyl)methyl]am...)
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50262290(4-[(3S,6S,9S,12S,20S)-6-(3-{[amino(iminiumyl)methy...)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50106479(FGGFTGARKSARK | H-FGGFTGARKSARK-NH2 | NC(1-13)NH2 ...)
Affinity DataKi:  0.350nMAssay Description:Binding affinity to human NOP receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50262292([Asp6,Lys10]N/OFQ(1-13)NH2 | CHEMBL507269)
Affinity DataKi:  0.540nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50106479(FGGFTGARKSARK | H-FGGFTGARKSARK-NH2 | NC(1-13)NH2 ...)
Affinity DataKi:  0.620nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50106469(FGGFTCARKCARK | cyclo[Cys6,Cys10]N/OFQ(1-13)NH2 | ...)
Affinity DataKi:  0.830nMAssay Description:Binding affinity to human NOP receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNociceptin receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50262293([D-Asp7,Lys10]N/OFQ(1-13)NH2 | CHEMBL507653)
Affinity DataKi:  1.79nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed