Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 2892
TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25891((2S)-2-[(5-formyl-1H-pyrrol-2-yl)formamido]-3-meth...)
Affinity DataIC50: 25nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25890((2S)-2-[(5-formylthiophen-2-yl)formamido]-3-methyl...)
Affinity DataIC50: 85nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25892((2S)-2-[(4-formyl-1H-pyrrol-2-yl)formamido]-3-meth...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25889((2S)-2-[(5-formylfuran-2-yl)formamido]-3-methyl-N-...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25887((2S)-3-methyl-N-[(2S)-4-methyl-1-oxopentan-2-yl]-2...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25894((2S)-3-methyl-N-[(2S)-4-methyl-1-oxopentan-2-yl]-2...)
Affinity DataIC50: 110nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25886((2S)-2-(furan-2-ylformamido)-3-methyl-N-[(2S)-4-me...)
Affinity DataIC50: 135nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25895(methyl 5-{[(1S)-2-methyl-1-{[(2S)-4-methyl-1-oxope...)
Affinity DataIC50: 140nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25893((2S)-2-[(5-formyl-1-methyl-1H-pyrrol-2-yl)formamid...)
Affinity DataIC50: 150nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25893((2S)-2-[(5-formyl-1-methyl-1H-pyrrol-2-yl)formamid...)
Affinity DataIC50: 150nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25895(methyl 5-{[(1S)-2-methyl-1-{[(2S)-4-methyl-1-oxope...)
Affinity DataIC50: 290nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25891((2S)-2-[(5-formyl-1H-pyrrol-2-yl)formamido]-3-meth...)
Affinity DataIC50: 290nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25888((2S)-3-methyl-N-[(2S)-4-methyl-1-oxopentan-2-yl]-2...)
Affinity DataIC50: 315nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25894((2S)-3-methyl-N-[(2S)-4-methyl-1-oxopentan-2-yl]-2...)
Affinity DataIC50: 340nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25890((2S)-2-[(5-formylthiophen-2-yl)formamido]-3-methyl...)
Affinity DataIC50: 440nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25892((2S)-2-[(4-formyl-1H-pyrrol-2-yl)formamido]-3-meth...)
Affinity DataIC50: 530nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25888((2S)-3-methyl-N-[(2S)-4-methyl-1-oxopentan-2-yl]-2...)
Affinity DataIC50: 650nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25887((2S)-3-methyl-N-[(2S)-4-methyl-1-oxopentan-2-yl]-2...)
Affinity DataIC50: 680nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25886((2S)-2-(furan-2-ylformamido)-3-methyl-N-[(2S)-4-me...)
Affinity DataIC50: 790nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25889((2S)-2-[(5-formylfuran-2-yl)formamido]-3-methyl-N-...)
Affinity DataIC50: 960nMpH: 7.5 T: 2°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed