Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50026438
TargetCathepsin K(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252525(benzyl 1-(2-cyanopiperazin-1-yl)-3-methyl-1-oxobut...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human recombinant cathepsin KMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin K(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252522(2-(2-(3-cyanophenylamino)-3-methylbutanoyl)piperaz...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant cathepsin KMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin K(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252523(2-(2-(m-toluidino)-3-methylbutanoyl)piperazine-1-c...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant cathepsin KMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252525(benzyl 1-(2-cyanopiperazin-1-yl)-3-methyl-1-oxobut...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin K(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252488(2-(2-(3-chlorophenylamino)-3-methylbutanoyl)pipera...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant cathepsin KMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252489(2-(3-methyl-2-(3-(trifluoromethyl)phenylamino)buta...)
Affinity DataIC50: 23nMAssay Description:Inhibition of human recombinant cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin K(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252489(2-(3-methyl-2-(3-(trifluoromethyl)phenylamino)buta...)
Affinity DataIC50: 23nMAssay Description:Inhibition of human recombinant cathepsin KMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin K(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252487(2-(2-(4-chlorophenylamino)-3-methylbutanoyl)pipera...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human recombinant cathepsin KMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin K(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252486(2-(3-methyl-2-(phenylamino)butanoyl)piperazine-1-c...)
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant cathepsin KMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252523(2-(2-(m-toluidino)-3-methylbutanoyl)piperazine-1-c...)
Affinity DataIC50: 32nMAssay Description:Inhibition of human recombinant cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252488(2-(2-(3-chlorophenylamino)-3-methylbutanoyl)pipera...)
Affinity DataIC50: 32nMAssay Description:Inhibition of human recombinant cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252524(tert-butyl 1-(2-cyanopiperazin-1-yl)-3-methyl-1-ox...)
Affinity DataIC50: 38nMAssay Description:Inhibition of human recombinant cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252522(2-(2-(3-cyanophenylamino)-3-methylbutanoyl)piperaz...)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProcathepsin L(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252489(2-(3-methyl-2-(3-(trifluoromethyl)phenylamino)buta...)
Affinity DataIC50: 48nMAssay Description:Inhibition of human recombinant cathepsin LMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252486(2-(3-methyl-2-(phenylamino)butanoyl)piperazine-1-c...)
Affinity DataIC50: 53nMAssay Description:Inhibition of human recombinant cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin K(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252524(tert-butyl 1-(2-cyanopiperazin-1-yl)-3-methyl-1-ox...)
Affinity DataIC50: 55nMAssay Description:Inhibition of human recombinant cathepsin KMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252487(2-(2-(4-chlorophenylamino)-3-methylbutanoyl)pipera...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProcathepsin L(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252524(tert-butyl 1-(2-cyanopiperazin-1-yl)-3-methyl-1-ox...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human recombinant cathepsin LMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProcathepsin L(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252525(benzyl 1-(2-cyanopiperazin-1-yl)-3-methyl-1-oxobut...)
Affinity DataIC50: 145nMAssay Description:Inhibition of human recombinant cathepsin LMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProcathepsin L(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252488(2-(2-(3-chlorophenylamino)-3-methylbutanoyl)pipera...)
Affinity DataIC50: 240nMAssay Description:Inhibition of human recombinant cathepsin LMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProcathepsin L(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252523(2-(2-(m-toluidino)-3-methylbutanoyl)piperazine-1-c...)
Affinity DataIC50: 355nMAssay Description:Inhibition of human recombinant cathepsin LMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProcathepsin L(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252487(2-(2-(4-chlorophenylamino)-3-methylbutanoyl)pipera...)
Affinity DataIC50: 610nMAssay Description:Inhibition of human recombinant cathepsin LMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProcathepsin L(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252486(2-(3-methyl-2-(phenylamino)butanoyl)piperazine-1-c...)
Affinity DataIC50: 625nMAssay Description:Inhibition of human recombinant cathepsin LMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProcathepsin L(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50252522(2-(2-(3-cyanophenylamino)-3-methylbutanoyl)piperaz...)
Affinity DataIC50: 730nMAssay Description:Inhibition of human recombinant cathepsin LMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed