Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50026375
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243356(N-[3,5-Bis(trifluoromethyl)benzyl]-N-methyl-5-phen...)
Affinity DataIC50: 4.30nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243233(N-[3,5-Bis(trifluoromethyl)benzyl]-N-methyl-5-phen...)
Affinity DataIC50: 9nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243449(N-[3,5-Bis(trifluoromethyl)benzyl]-5-(4-fluorophen...)
Affinity DataIC50: 21nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243403(N-[3,5-Bis(trifluoromethyl)benzyl]-N-methyl-5-phen...)
Affinity DataIC50: 26nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243307(N-[3,5-Bis(trifluoromethyl)benzyl]-N-methyl-5-phen...)
Affinity DataIC50: 36nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243309(N-[3,5-Bis(trifluoromethyl)benzyl]-N-methyl-5-phen...)
Affinity DataIC50: 38nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243405(N-[3,5-Bis(trifluoromethyl)benzyl]-N-methyl-5-(4-m...)
Affinity DataIC50: 55nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243355(N-[3,5-Bis(trifluoromethyl)benzyl]-5-phenylimidazo...)
Affinity DataIC50: 146nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243448(N-[3,5-Bis(trifluoromethyl)benzyl]-5-(4-fluorophen...)
Affinity DataIC50: 235nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243234(N-[3,5-Bis(trifluoromethyl)benzyl]-5-phenyltetrazo...)
Affinity DataIC50: 311nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243235(N-[3,5-Bis(trifluoromethyl)benzyl]-5-phenylpyrrolo...)
Affinity DataIC50: 390nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243404(N-[3,5-Bis(trifluoromethyl)benzyl]-5-(4-methylphen...)
Affinity DataIC50: 401nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243357(N-[3,5-Bis(trifluoromethyl)benzyl]-5-phenyl[1,2,4]...)
Affinity DataIC50: 542nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243451(N-(3,5-dimethoxybenzyl)-5-phenyltetrazolo[1,5-a]qu...)
Affinity DataIC50: 780nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243308(N-[3,5-Bis(trifluoromethyl)benzyl]-5-phenylimidazo...)
Affinity DataIC50: 1.23E+3nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50243450(N-(2-Methoxybenzyl)-5-phenyltetrazolo[1,5-a]quinol...)
Affinity DataIC50: 2.75E+3nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed