Compile Data Set for Download or QSAR
Report error Found 106 Enz. Inhib. hit(s) with all data for entry = 50026322
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243780(2-(dimethylamino)-1-(4-(6-phenyl-7-(4-((4-(5-(pyri...)
Affinity DataIC50: 3nMAssay Description:Inhibition of Akt1 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(N,N-dimethyl-2-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2...)
Affinity DataIC50: 4nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(N,N-dimethyl-2-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2...)
Affinity DataIC50: 4nMAssay Description:Inhibition of Akt2 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243777(1-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50: 5nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243776(2-(1H-imidazol-1-yl)-6-phenyl-7-(4-((4-(5-(pyridin...)
Affinity DataIC50: 5nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243764(2-morpholino-6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4...)
Affinity DataIC50: 5nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243780(2-(dimethylamino)-1-(4-(6-phenyl-7-(4-((4-(5-(pyri...)
Affinity DataIC50: 6nMAssay Description:Inhibition of Akt2 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243783(2-(4-(1-methylazetidin-3-yl)piperazin-1-yl)-6-phen...)
Affinity DataIC50: 6nMAssay Description:Inhibition of Akt1 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24880(N-methyl-6-phenyl-7-[4-({4-[5-(pyridin-2-yl)-4H-1,...)
Affinity DataIC50: 6nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243780(2-(dimethylamino)-1-(4-(6-phenyl-7-(4-((4-(5-(pyri...)
Affinity DataIC50: 6nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243778(2-(4-(methylsulfonyl)piperazin-1-yl)-6-phenyl-7-(4...)
Affinity DataIC50: 7nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243765(1-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4-tr...)
Affinity DataIC50: 7nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243769(2-((R)-3-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(...)
Affinity DataIC50: 8nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243782(2-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50: 9nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243771(2-(4-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(5-(p...)
Affinity DataIC50: 9nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243783(2-(4-(1-methylazetidin-3-yl)piperazin-1-yl)-6-phen...)
Affinity DataIC50: 9nMAssay Description:Inhibition of Akt2 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(N,N-dimethyl-2-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2...)
Affinity DataIC50: 10nMAssay Description:Inhibition of Akt1 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243775(N,N-dimethyl-1-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl...)
Affinity DataIC50: 10nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243783(2-(4-(1-methylazetidin-3-yl)piperazin-1-yl)-6-phen...)
Affinity DataIC50: 12nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243779(N,N-dimethyl-4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl...)
Affinity DataIC50: 13nMAssay Description:Inhibition of Akt1 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243777(1-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50: 15nMAssay Description:Inhibition of Akt1 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24867(CHEMBL252456 | 1-(2-aminophenyl)-3-[({4-[2-(methyl...)
Affinity DataIC50: 15nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243777(1-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50: 16nMAssay Description:Inhibition of Akt2 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243782(2-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50: 17nMAssay Description:Inhibition of Akt1 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243765(1-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4-tr...)
Affinity DataIC50: 17nMAssay Description:Inhibition of Akt1 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243770(2-((S)-3-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(...)
Affinity DataIC50: 17nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243779(N,N-dimethyl-4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl...)
Affinity DataIC50: 18nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243763(6-phenyl-2-(piperidin-1-yl)-7-(4-((4-(5-(pyridin-2...)
Affinity DataIC50: 18nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243764(2-morpholino-6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4...)
Affinity DataIC50: 19nMAssay Description:Inhibition of Akt1 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243780(2-(dimethylamino)-1-(4-(6-phenyl-7-(4-((4-(5-(pyri...)
Affinity DataIC50: 19nMAssay Description:Inhibition of Akt2 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243781(2-(5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)...)
Affinity DataIC50: 19nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243778(2-(4-(methylsulfonyl)piperazin-1-yl)-6-phenyl-7-(4...)
Affinity DataIC50: 20nMAssay Description:Inhibition of Akt1 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24880(N-methyl-6-phenyl-7-[4-({4-[5-(pyridin-2-yl)-4H-1,...)
Affinity DataIC50: 20nMAssay Description:Inhibition of Akt1 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243762(2-(3,3-difluoropyrrolidin-1-yl)-6-phenyl-7-(4-((4-...)
Affinity DataIC50: 20nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243775(N,N-dimethyl-1-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl...)
Affinity DataIC50: 22nMAssay Description:Inhibition of Akt2 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243778(2-(4-(methylsulfonyl)piperazin-1-yl)-6-phenyl-7-(4...)
Affinity DataIC50: 23nMAssay Description:Inhibition of Akt2 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243775(N,N-dimethyl-1-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl...)
Affinity DataIC50: 23nMAssay Description:Inhibition of Akt1 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243769(2-((R)-3-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(...)
Affinity DataIC50: 25nMAssay Description:Inhibition of Akt2 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243774((2R)-4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2...)
Affinity DataIC50: 25nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243771(2-(4-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(5-(p...)
Affinity DataIC50: 27nMAssay Description:Inhibition of Akt2 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243783(2-(4-(1-methylazetidin-3-yl)piperazin-1-yl)-6-phen...)
Affinity DataIC50: 27nMAssay Description:Inhibition of Akt2 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243766(2-((2S,6R)-2,6-dimethylmorpholino)-6-phenyl-7-(4-(...)
Affinity DataIC50: 28nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243772(2-((2R,5S)-2,5-dimethylpiperazin-1-yl)-6-phenyl-7-...)
Affinity DataIC50: 29nMAssay Description:Inhibition of Akt2 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243782(2-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50: 31nMAssay Description:Inhibition of Akt2 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243776(2-(1H-imidazol-1-yl)-6-phenyl-7-(4-((4-(5-(pyridin...)
Affinity DataIC50: 35nMAssay Description:Inhibition of Akt1 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243771(2-(4-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(5-(p...)
Affinity DataIC50: 36nMAssay Description:Inhibition of Akt1 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243769(2-((R)-3-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(...)
Affinity DataIC50: 36nMAssay Description:Inhibition of Akt1 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243763(6-phenyl-2-(piperidin-1-yl)-7-(4-((4-(5-(pyridin-2...)
Affinity DataIC50: 36nMAssay Description:Inhibition of Akt1 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243767(2-(1,1-Dioxo-1lambda6-thiomorpholin-4-yl)-6-phenyl...)
Affinity DataIC50: 38nMAssay Description:Inhibition of Akt1 phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(N,N-dimethyl-2-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2...)
Affinity DataIC50: 39nMAssay Description:Inhibition of Akt2 phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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