Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 3585
TargetGlycogen synthase kinase-3 beta(Human)
University of Pennsylvania

LigandPNGBDBM36523(DW12)
Affinity DataIC50: 1.40nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36525(EAd125)
Affinity DataIC50: 40nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Pennsylvania

LigandPNGBDBM36522(HB12)
Affinity DataIC50: 50nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36525(EAd125)
Affinity DataIC50: 180nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36524(DW12Me)
Affinity DataIC50: 500nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Pennsylvania

LigandPNGBDBM36525(EAd125)
Affinity DataIC50: 700nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36523(DW12)
Affinity DataIC50: 750nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36522(HB12)
Affinity DataIC50: 1.00E+3nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Pennsylvania

LigandPNGBDBM36524(DW12Me)
Affinity DataIC50: 1.00E+3nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Pennsylvania

LigandPNGBDBM36525(EAd125)
Affinity DataIC50: 4.00E+3nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed