Compile Data Set for Download or QSAR
Report error Found 57 Enz. Inhib. hit(s) with all data for entry = 2723
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23843(5,16,25-trimethoxy-14-oxapentacyclo[20.2.2.2^{10,1...)
Affinity DataIC50: 2.00E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23844(16,25-dimethoxy-14-oxapentacyclo[20.2.2.2^{10,13}....)
Affinity DataIC50: 2.20E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23848(25-methoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1^{15...)
Affinity DataIC50: 2.50E+3nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23842(2-[2,6-bis(propan-2-yl)phenyl]-3-sulfanylidene-2,3...)
Affinity DataIC50: 3.10E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23853(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 3.20E+3nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23845(5,16-dimethoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1...)
Affinity DataIC50: 3.60E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23850(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 4.40E+3nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM19992(2-{3-[3-({[2-chloro-3-(trifluoromethyl)phenyl]meth...)
Affinity DataIC50: 4.80E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23839(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 4.90E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM23850(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 4.90E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM23851(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 5.10E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23852(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 5.70E+3nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23839(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 6.60E+3nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23849(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 6.60E+3nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23854(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 7.10E+3nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23853(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 7.30E+3nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23847(16-methoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1^{15...)
Affinity DataIC50: 7.60E+3nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23850(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 7.60E+3nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM23842(2-[2,6-bis(propan-2-yl)phenyl]-3-sulfanylidene-2,3...)
Affinity DataIC50: 8.00E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23851(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 8.40E+3nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM23849(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 8.60E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23840(2-[2-(2-phenylethyl)phenyl]-2,3-dihydro-1H-isoindo...)
Affinity DataIC50: 9.80E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM23839(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 9.90E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23851(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 1.00E+4nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23848(25-methoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1^{15...)
Affinity DataIC50: 1.10E+4nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23844(16,25-dimethoxy-14-oxapentacyclo[20.2.2.2^{10,13}....)
Affinity DataIC50: 1.20E+4nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23841(CHEMBL245943 | 2-(2-hexylphenyl)-2,3-dihydro-1H-is...)
Affinity DataIC50: 1.30E+4nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23849(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 1.30E+4nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23843(5,16,25-trimethoxy-14-oxapentacyclo[20.2.2.2^{10,1...)
Affinity DataIC50: 1.40E+4nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23852(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 1.40E+4nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM23852(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 1.50E+4nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM23840(2-[2-(2-phenylethyl)phenyl]-2,3-dihydro-1H-isoindo...)
Affinity DataIC50: 1.62E+4nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23842(2-[2,6-bis(propan-2-yl)phenyl]-3-sulfanylidene-2,3...)
Affinity DataIC50: 1.80E+4nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM23854(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 1.80E+4nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM23853(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 1.90E+4nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM19459(Prunetol | Genisteol | CHEMBL44 | US8552057, 2 | c...)
Affinity DataIC50: 2.20E+4nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM23841(CHEMBL245943 | 2-(2-hexylphenyl)-2,3-dihydro-1H-is...)
Affinity DataIC50: 2.47E+4nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM23846(5,25-dimethoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1...)
Affinity DataIC50: 2.50E+4nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23845(5,16-dimethoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1...)
Affinity DataIC50: 2.60E+4nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM23846(5,25-dimethoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1...)
Affinity DataIC50: 3.00E+4nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
University of Tokyo

LigandPNGBDBM19459(Prunetol | Genisteol | CHEMBL44 | US8552057, 2 | c...)
Affinity DataIC50: 3.10E+4nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM23845(5,16-dimethoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1...)
Affinity DataIC50: 4.00E+4nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23847(16-methoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1^{15...)
Affinity DataIC50: 4.10E+4nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM23844(16,25-dimethoxy-14-oxapentacyclo[20.2.2.2^{10,13}....)
Affinity DataIC50: 4.20E+4nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23840(2-[2-(2-phenylethyl)phenyl]-2,3-dihydro-1H-isoindo...)
Affinity DataIC50: 4.40E+4nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23846(5,25-dimethoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1...)
Affinity DataIC50: 4.60E+4nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM23843(5,16,25-trimethoxy-14-oxapentacyclo[20.2.2.2^{10,1...)
Affinity DataIC50: 4.90E+4nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23841(CHEMBL245943 | 2-(2-hexylphenyl)-2,3-dihydro-1H-is...)
Affinity DataIC50: 6.50E+4nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL32(Baker's yeast)
University of Tokyo

LigandPNGBDBM23848(25-methoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1^{15...)
Affinity DataIC50: 6.70E+4nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
University of Tokyo

LigandPNGBDBM23854(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50: 7.70E+4nMAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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