Compile Data Set for Download or QSAR
Report error Found 276 Enz. Inhib. hit(s) with all data for entry = 50038071
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371255(CHEMBL1203953)
Affinity DataIC50: 0.180nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232520((2R)-4-oxo-4-[3-(trifluoromethyl)-8-[2-(trifluorom...)
Affinity DataIC50: 0.310nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232520((2R)-4-oxo-4-[3-(trifluoromethyl)-8-[2-(trifluorom...)
Affinity DataIC50: 0.310nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232506(2-[7-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50: 0.320nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232518((2R)-4-oxo-4-[8-(pyridin-2-ylmethyl)-3-(trifluorom...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232518((2R)-4-oxo-4-[8-(pyridin-2-ylmethyl)-3-(trifluorom...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232503((2R)-4-[8-(4-methoxybenzyl)-3-(trifluoromethyl)-5,...)
Affinity DataIC50: 0.430nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232503((2R)-4-[8-(4-methoxybenzyl)-3-(trifluoromethyl)-5,...)
Affinity DataIC50: 0.430nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232501((2R)-4-[8-(2-fluorobenzyl)-3-(trifluoromethyl)-5,6...)
Affinity DataIC50: 0.460nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232501((2R)-4-[8-(2-fluorobenzyl)-3-(trifluoromethyl)-5,6...)
Affinity DataIC50: 0.460nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232506(2-[7-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232506(2-[7-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232510((2R)-4-[8-benzyl-3-(trifluoromethyl)-5,6-dihydro[1...)
Affinity DataIC50: 0.660nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232510((2R)-4-[8-benzyl-3-(trifluoromethyl)-5,6-dihydro[1...)
Affinity DataIC50: 0.660nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232507(2-[7-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232507(2-[7-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232502((2R)-4-[(8S)-8-methyl-3-(trifluoromethyl)-5,6-dihy...)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232511((2R)-4-[8-ethyl-3-(trifluoromethyl)-5,6-dihydro[1,...)
Affinity DataIC50: 5nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232511((2R)-4-[8-ethyl-3-(trifluoromethyl)-5,6-dihydro[1,...)
Affinity DataIC50: 5nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232508((2R)-4-[8-(2,2,2-trifluoroethyl)-3-(trifluoromethy...)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232508((2R)-4-[8-(2,2,2-trifluoroethyl)-3-(trifluoromethy...)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232519((2R)-4-[8-[3,5-bis(trifluoromethyl)benzyl]-3-(trif...)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232519((2R)-4-[8-[3,5-bis(trifluoromethyl)benzyl]-3-(trif...)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232504((2R)-4-[5,8-dimethyl-3-(trifluoromethyl)-5,6-dihyd...)
Affinity DataIC50: 11nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232502((2R)-4-[(8S)-8-methyl-3-(trifluoromethyl)-5,6-dihy...)
Affinity DataIC50: 11nMAssay Description:Inhibition of mouse DPP4 at 1 mg/kgMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232504((2R)-4-[5,8-dimethyl-3-(trifluoromethyl)-5,6-dihyd...)
Affinity DataIC50: 11nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232504((2R)-4-[5,8-dimethyl-3-(trifluoromethyl)-5,6-dihyd...)
Affinity DataIC50: 12nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM11162(Triazolopiperazine Analogue 1 | (3R)-3-amino-1-[3-...)
Affinity DataIC50: 18nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232514((2R)-4-[8-allyl-3-(trifluoromethyl)-5,6-dihydro[[1...)
Affinity DataIC50: 32nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232514((2R)-4-[8-allyl-3-(trifluoromethyl)-5,6-dihydro[[1...)
Affinity DataIC50: 32nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232521((2R)-4-[(6R)-6-methyl-3-(trifluoromethyl)-5,6-dihy...)
Affinity DataIC50: 42nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM11162(Triazolopiperazine Analogue 1 | (3R)-3-amino-1-[3-...)
Affinity DataIC50: 69nMAssay Description:Inhibition of mouse DPP4 at 3 mg/kgMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232502((2R)-4-[(8S)-8-methyl-3-(trifluoromethyl)-5,6-dihy...)
Affinity DataIC50: 88nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232506(2-[7-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50: 90nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232500(((2R)-4-[(6S)-6-methyl-3-(trifluoromethyl)-5,6-dih...)
Affinity DataIC50: 91nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232505((2R)-4-[5,5-dimethyl-3-(trifluoromethyl)-5,6-dihyd...)
Affinity DataIC50: 92nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232512((2R)-4-[(8S)-8-(4-fluorobenzyl)-3-(trifluoromethyl...)
Affinity DataIC50: 116nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50151843((R)-3-Amino-1-((R)-2-benzyl-piperazin-1-yl)-4-(2-f...)
Affinity DataIC50: 139nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232524((2R)-4-[8,8-dimethyl-3-(trifluoromethyl)-5,6-dihyd...)
Affinity DataIC50: 175nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232504((2R)-4-[5,8-dimethyl-3-(trifluoromethyl)-5,6-dihyd...)
Affinity DataIC50: 209nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371255(CHEMBL1203953)
Affinity DataIC50: 332nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232503((2R)-4-[8-(4-methoxybenzyl)-3-(trifluoromethyl)-5,...)
Affinity DataIC50: 367nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232510((2R)-4-[8-benzyl-3-(trifluoromethyl)-5,6-dihydro[1...)
Affinity DataIC50: 622nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232506(2-[7-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50: 628nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232506(2-[7-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50: 628nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232501((2R)-4-[8-(2-fluorobenzyl)-3-(trifluoromethyl)-5,6...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232508((2R)-4-[8-(2,2,2-trifluoroethyl)-3-(trifluoromethy...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50151819((R)-3-Amino-4-(2-fluoro-phenyl)-1-piperazin-1-yl-b...)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232518((2R)-4-oxo-4-[8-(pyridin-2-ylmethyl)-3-(trifluorom...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50232524((2R)-4-[8,8-dimethyl-3-(trifluoromethyl)-5,6-dihyd...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
Displayed 1 to 50 (of 276 total ) | Next | Last >>
Jump to: