Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50022181
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM19331(CHEMBL266063 | N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(...)
Affinity DataIC50: 0.600nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232281((R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-t...)
Affinity DataIC50: 0.700nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232297((R)-N-((4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2...)
Affinity DataIC50: 1.10nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM19331(CHEMBL266063 | N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(...)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at GHSR1a expressed in CHO cells assessed as accumulation of intracellular calcium levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232283((R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethox...)
Affinity DataIC50: 1.80nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232270((R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyben...)
Affinity DataIC50: 1.90nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232266((R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-t...)
Affinity DataIC50: 3nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50208689((R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(3-methoxyb...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at GHSR1a expressed in CHO cells assessed as accumulation of intracellular calcium levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232295((R)-N-((4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2...)
Affinity DataIC50: 5nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM19312(CHEMBL253126 | (2S)-N-[(1R)-1-{4-[(2,4-dimethoxyph...)
Affinity DataIC50: 5.60nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM19294(CHEMBL374643 | 2-amino-N-[(1R)-2-(1H-indol-3-yl)-1...)
Affinity DataIC50: 6nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232274((R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyben...)
Affinity DataIC50: 7.90nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232264(N-((R)-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-t...)
Affinity DataIC50: 11nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232263((R)-N-((4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2...)
Affinity DataIC50: 11.8nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232268((R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-t...)
Affinity DataIC50: 14nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232263((R)-N-((4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at GHSR1a expressed in CHO cells assessed as accumulation of intracellular calcium levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50208689((R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(3-methoxyb...)
Affinity DataIC50: 18nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232293((R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethox...)
Affinity DataIC50: 18.5nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232286((R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-t...)
Affinity DataIC50: 29nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232277(N-((R)-(4-(2,4-dimethoxyphenyl)-5-phenethyl-4H-1,2...)
Affinity DataIC50: 33nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232269((R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethox...)
Affinity DataIC50: 34nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232279((R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(4-ethylpheny...)
Affinity DataIC50: 49nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232285((R)-N-((4-(4-ethylbenzyl)-5-phenethyl-4H-1,2,4-tri...)
Affinity DataIC50: 51nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232300((R)-N-((4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2...)
Affinity DataIC50: 58nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232292(N-((R)-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2...)
Affinity DataIC50: 60nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232276((R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-benzyl-4H-1,2...)
Affinity DataIC50: 61nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232294((R)-N-((4-(4-ethylbenzyl)-5-phenethyl-4H-1,2,4-tri...)
Affinity DataIC50: 67nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232291((R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyben...)
Affinity DataIC50: 76nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232298((R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-t...)
Affinity DataIC50: 80nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232282((R)-N-((4-(4-ethylbenzyl)-5-phenethyl-4H-1,2,4-tri...)
Affinity DataIC50: 89nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232278((R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(4-ethylpheny...)
Affinity DataIC50: 96nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232288((R)-N-((1H-indol-3-yl)(5-phenethyl-4-phenyl-4H-1,2...)
Affinity DataIC50: 105nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232272(N-((R)-(5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethox...)
Affinity DataIC50: 108nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232296((R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethox...)
Affinity DataIC50: 112nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232287(N-((R)-(4-(2,4-dimethoxyphenyl)-5-phenethyl-4H-1,2...)
Affinity DataIC50: 120nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232289((1S,2R)-N-((R)-(5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-...)
Affinity DataIC50: 140nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232290((R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-phenyl-4H-1,2...)
Affinity DataIC50: 160nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232267((R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-t...)
Affinity DataIC50: 177nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232280((R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-t...)
Affinity DataIC50: 220nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232299((R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-t...)
Affinity DataIC50: 270nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232271(N-((R)-(4-(2,4-dimethoxyphenyl)-5-phenethyl-4H-1,2...)
Affinity DataIC50: 300nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232284((R)-N-((4-(4-ethylbenzyl)-5-phenethyl-4H-1,2,4-tri...)
Affinity DataIC50: 480nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232265((R)-N-((1H-indol-3-yl)(5-phenethyl-4-phenyl-4H-1,2...)
Affinity DataIC50: 700nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232273((R)-N-((4-(4-ethylbenzyl)-5-phenethyl-4H-1,2,4-tri...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50232275((R)-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of 125I]-His9-ghrelin from human GHSR1a expressed in LLCPK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed