Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50003947
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477891(CHEMBL401641)
Affinity DataEC50:  132nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477901(CHEMBL437201)
Affinity DataEC50:  0.676nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477900(CHEMBL437199)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50412707(CHEMBL230333)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477899(CHEMBL438162)
Affinity DataEC50:  0.646nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477898(CHEMBL441576)
Affinity DataEC50:  0.708nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477897(CHEMBL427638)
Affinity DataEC50:  8.10nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477896(CHEMBL268436)
Affinity DataEC50:  8.30nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477895(CHEMBL409981)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477894(CHEMBL398483)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477893(CHEMBL398524)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477892(CHEMBL411392)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477880(CHEMBL430024)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477890(CHEMBL267266)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477889([2Nal2]hNPS)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477888(CHEMBL411571)
Affinity DataEC50:  34nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477887(CHEMBL437389)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477886(CHEMBL409555)
Affinity DataEC50:  15nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477885(CHEMBL252537)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477884(CHEMBL267034)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477883(CHEMBL400369)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477882(CHEMBL413849)
Affinity DataEC50:  4.20nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477881(CHEMBL2372117)
Affinity DataEC50:  11nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed