Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50038257
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231845(N-(3-chloro-4-(4-ethylpiperazin-1-yl)phenyl)-3-cyc...)
Affinity DataIC50: 440nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373835(CHEMBL256202)
Affinity DataIC50: 490nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373841(CHEMBL270580)
Affinity DataIC50: 580nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231845(N-(3-chloro-4-(4-ethylpiperazin-1-yl)phenyl)-3-cyc...)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373834(CHEMBL255169)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373836(CHEMBL271704)
Affinity DataIC50: 1.15E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231845(N-(3-chloro-4-(4-ethylpiperazin-1-yl)phenyl)-3-cyc...)
Affinity DataIC50: 3.10E+3nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373832(CHEMBL429780)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231845(N-(3-chloro-4-(4-ethylpiperazin-1-yl)phenyl)-3-cyc...)
Affinity DataIC50: 3.50E+3nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373837(CHEMBL429320)
Affinity DataIC50: 4.60E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231856(N-(3-chloro-4-(4-ethylpiperazin-1-yl)phenyl)benzam...)
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373835(CHEMBL256202)
Affinity DataIC50: 5.10E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373839(CHEMBL438706)
Affinity DataIC50: 5.60E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373834(CHEMBL255169)
Affinity DataIC50: 7.60E+3nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373841(CHEMBL270580)
Affinity DataIC50: 7.90E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373836(CHEMBL271704)
Affinity DataIC50: 1.30E+4nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373834(CHEMBL255169)
Affinity DataIC50: 1.80E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373838(CHEMBL258335)
Affinity DataIC50: 1.88E+4nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373836(CHEMBL271704)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373836(CHEMBL271704)
Affinity DataIC50: 2.40E+4nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373836(CHEMBL271704)
Affinity DataIC50: 2.90E+4nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373834(CHEMBL255169)
Affinity DataIC50: 5.20E+4nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231856(N-(3-chloro-4-(4-ethylpiperazin-1-yl)phenyl)benzam...)
Affinity DataIC50: 6.60E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373834(CHEMBL255169)
Affinity DataIC50: 7.00E+4nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373839(CHEMBL438706)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373833(CHEMBL404874)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373840(CHEMBL258281)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373832(CHEMBL429780)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373840(CHEMBL258281)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373837(CHEMBL429320)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231856(N-(3-chloro-4-(4-ethylpiperazin-1-yl)phenyl)benzam...)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373837(CHEMBL429320)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231845(N-(3-chloro-4-(4-ethylpiperazin-1-yl)phenyl)-3-cyc...)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373832(CHEMBL429780)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373838(CHEMBL258335)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373840(CHEMBL258281)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373837(CHEMBL429320)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373839(CHEMBL438706)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373833(CHEMBL404874)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373838(CHEMBL258335)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373840(CHEMBL258281)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373833(CHEMBL404874)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373837(CHEMBL429320)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373838(CHEMBL258335)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373839(CHEMBL438706)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373840(CHEMBL258281)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373835(CHEMBL256202)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231856(N-(3-chloro-4-(4-ethylpiperazin-1-yl)phenyl)benzam...)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373833(CHEMBL404874)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Vanderbilt Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373835(CHEMBL256202)
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
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