Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50003944
TargetAmyloid-beta precursor protein(Human)
National Institute of Mental Health

Curated by ChEMBL
LigandPNGBDBM50129793(N-methyl-[11C]2-(40-methylaminophenyl)-6-hydroxy b...)
Affinity DataKd:  7.20nMAssay Description:Binding affinity to beta amyloid plaque in human Alzheimer's disease brain tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
National Institute of Mental Health

Curated by ChEMBL
LigandPNGBDBM50477824(CHEMBL252766)
Affinity DataKi:  7.90nMAssay Description:Binding affinity to beta amyloid plaque in human Alzheimer's disease brain tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
National Institute of Mental Health

Curated by ChEMBL
LigandPNGBDBM50122787(4-(6-iodoimidazo[1,2-a]pyridin-2-yl)-N,N-dimethyla...)
Affinity DataKi:  9nMAssay Description:Binding affinity to beta amyloid plaque in human Alzheimer's disease brain tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
National Institute of Mental Health

Curated by ChEMBL
LigandPNGBDBM50477826(CHEMBL252765)
Affinity DataKi:  80nMAssay Description:Binding affinity to beta amyloid plaque in human Alzheimer's disease brain tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
National Institute of Mental Health

Curated by ChEMBL
LigandPNGBDBM50477823(CHEMBL252969)
Affinity DataKi:  205nMAssay Description:Binding affinity to beta amyloid plaque in human Alzheimer's disease brain tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
National Institute of Mental Health

Curated by ChEMBL
LigandPNGBDBM50477825(CHEMBL254850)
Affinity DataKi:  377nMAssay Description:Binding affinity to beta amyloid plaque in human Alzheimer's disease brain tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed