Compile Data Set for Download or QSAR
Report error Found 100 Enz. Inhib. hit(s) with all data for entry = 50021901
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229206(N-(4-(trifluoromethylsulfonamido)benzyl)-4-methyl-...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229219(4'-chloro-biphenyl-4-carboxylic acid 4-trifluorome...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229217(N-(4-(2,2,2-trifluoroacetamido)benzyl)-4-methyl-2-...)
Affinity DataEC50:  450nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229216(N-(4-(2-hydroxy-3,4-dioxocyclobut-1-enyl)benzyl)-4...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28706(CHEMBL219586 | 2-methyl-2-{4-[({4-methyl-2-[4-(tri...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229219(4'-chloro-biphenyl-4-carboxylic acid 4-trifluorome...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229212(N-(4-(propan-2-ylsulfonamido)benzyl)-4-methyl-2-(4...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229227(2-(4-((4-(5-(methoxymethyl)-1,2,4-oxadiazol-3-yl)b...)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229208(N-(4-(2,2,2-trifluoroethylsulfonamido)benzyl)-4-me...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229205(N-(4-((trifluoromethylsulfonamido)methyl)benzyl)-4...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229209(N-(4-(4-methylphenylsulfonamido)benzyl)-4-methyl-2...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229212(N-(4-(propan-2-ylsulfonamido)benzyl)-4-methyl-2-(4...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229220(N-(4-(methylsulfonamido)benzyl)-4-methyl-2-(4-(tri...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229216(N-(4-(2-hydroxy-3,4-dioxocyclobut-1-enyl)benzyl)-4...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229222(N-(4-(butylsulfonamido)benzyl)-4-methyl-2-(4-(trif...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229225(2-(4-((5-methoxybenzo[b]thiophene-2-carboxamido)me...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229215(N-(4-((2H-tetrazol-5-yl)methoxy)benzyl)-4-methyl-2...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229211(N-(4-(2-methyl-1-oxo-1-(trifluoromethylsulfonamido...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229211(N-(4-(2-methyl-1-oxo-1-(trifluoromethylsulfonamido...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229221(2-(4'-chloro-biphenyl-4-yl)-N-(4-trifluoromethanes...)
Affinity DataEC50:  340nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229220(N-(4-(methylsulfonamido)benzyl)-4-methyl-2-(4-(tri...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229216(N-(4-(2-hydroxy-3,4-dioxocyclobut-1-enyl)benzyl)-4...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229206(N-(4-(trifluoromethylsulfonamido)benzyl)-4-methyl-...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229212(N-(4-(propan-2-ylsulfonamido)benzyl)-4-methyl-2-(4...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229209(N-(4-(4-methylphenylsulfonamido)benzyl)-4-methyl-2...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229216(N-(4-(2-hydroxy-3,4-dioxocyclobut-1-enyl)benzyl)-4...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229205(N-(4-((trifluoromethylsulfonamido)methyl)benzyl)-4...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229220(N-(4-(methylsulfonamido)benzyl)-4-methyl-2-(4-(tri...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28706(CHEMBL219586 | 2-methyl-2-{4-[({4-methyl-2-[4-(tri...)
Affinity DataEC50:  9.70E+3nMAssay Description:Agonist activity at mouse PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229206(N-(4-(trifluoromethylsulfonamido)benzyl)-4-methyl-...)
Affinity DataEC50:  600nMAssay Description:Agonist activity at mouse PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229216(N-(4-(2-hydroxy-3,4-dioxocyclobut-1-enyl)benzyl)-4...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229222(N-(4-(butylsulfonamido)benzyl)-4-methyl-2-(4-(trif...)
Affinity DataEC50:  6.70E+3nMAssay Description:Agonist activity at mouse PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229222(N-(4-(butylsulfonamido)benzyl)-4-methyl-2-(4-(trif...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28706(CHEMBL219586 | 2-methyl-2-{4-[({4-methyl-2-[4-(tri...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229205(N-(4-((trifluoromethylsulfonamido)methyl)benzyl)-4...)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229222(N-(4-(butylsulfonamido)benzyl)-4-methyl-2-(4-(trif...)
Affinity DataEC50:  320nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229220(N-(4-(methylsulfonamido)benzyl)-4-methyl-2-(4-(tri...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229209(N-(4-(4-methylphenylsulfonamido)benzyl)-4-methyl-2...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229215(N-(4-((2H-tetrazol-5-yl)methoxy)benzyl)-4-methyl-2...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229227(2-(4-((4-(5-(methoxymethyl)-1,2,4-oxadiazol-3-yl)b...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229215(N-(4-((2H-tetrazol-5-yl)methoxy)benzyl)-4-methyl-2...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229211(N-(4-(2-methyl-1-oxo-1-(trifluoromethylsulfonamido...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229224(2-(4-{[(4'-chloro-biphenyl-4-carbonyl)-amino]-meth...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229208(N-(4-(2,2,2-trifluoroethylsulfonamido)benzyl)-4-me...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at mouse PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229211(N-(4-(2-methyl-1-oxo-1-(trifluoromethylsulfonamido...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229206(N-(4-(trifluoromethylsulfonamido)benzyl)-4-methyl-...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28706(CHEMBL219586 | 2-methyl-2-{4-[({4-methyl-2-[4-(tri...)
Affinity DataEC50:  9.70E+3nMAssay Description:Agonist activity at human PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229226(N-(4-(trifluoromethylsulfonamido)benzyl)-4-(5-(met...)
Affinity DataEC50:  360nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229211(N-(4-(2-methyl-1-oxo-1-(trifluoromethylsulfonamido...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229219(4'-chloro-biphenyl-4-carboxylic acid 4-trifluorome...)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 100 total ) | Next | Last >>
Jump to: