Compile Data Set for Download or QSAR
Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 50038064
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227687(2-(2-(1-butyl-3-(4-isopropylphenyl)ureido)-2,3-dih...)
Affinity DataEC50:  260nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227691(2-(2-(3-(2,4-difluorophenyl)-1-heptylureido)-2,3-d...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227695((S)-2-(2-(1-heptyl-3-(4-(trifluoromethoxy)phenyl)u...)
Affinity DataEC50: >1.30E+4nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227696(2-methyl-2-(2-(3-(4-(trifluoromethoxy)phenyl)ureid...)
Affinity DataEC50:  96nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227689(2-methyl-2-(2-(1-(4,4,4-trifluorobutyl)-3-(4-(trif...)
Affinity DataEC50:  707nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227693(2-(2-(1-heptyl-3-(3-methoxyphenyl)ureido)-2,3-dihy...)
Affinity DataEC50:  1.11E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227692(2-(2-(1-isopentyl-3-(4-(trifluoromethoxy)phenyl)ur...)
Affinity DataEC50:  386nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227690(2-(2-(1-(2-methoxyethyl)-3-(4-(trifluoromethoxy)ph...)
Affinity DataEC50:  425nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227688(2-(2-(1-hexyl-3-(4-(trifluoromethoxy)phenyl)ureido...)
Affinity DataEC50:  166nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227694(2-(2-(3-(2-fluorophenyl)-1-heptylureido)-2,3-dihyd...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50371235(CIPROFIBRATE)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227685(2-(2-(1-hexyl-3-(4-(trifluoromethylthio)phenyl)ure...)
Affinity DataEC50:  249nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227686(2-(2-(1-isopropyl-3-(4-(trifluoromethoxy)phenyl)ur...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  190nMAssay Description:Agonist activity at PPARgamma expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM28799(2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)a...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at PPARgamma expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227680(2-(2-(1-heptyl-3-(2-(trifluoromethoxy)phenyl)ureid...)
Affinity DataEC50:  4.99E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227683(2-(2-(1-heptyl-3-(4-(trifluoromethoxy)phenyl)ureid...)
Affinity DataEC50:  294nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227684(2-(2-(1-heptyl-3-(2-(trifluoromethyl)phenyl)ureido...)
Affinity DataEC50:  6.39E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227701(2-methyl-2-(2-(1-octyl-3-(4-(trifluoromethoxy)phen...)
Affinity DataEC50:  1.03E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227700(2-(2-(1-heptyl-3-(4-methoxyphenyl)ureido)-2,3-dihy...)
Affinity DataEC50:  910nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227698(2-(2-(1-isobutyl-3-(4-(trifluoromethoxy)phenyl)ure...)
Affinity DataEC50:  2.34E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227699(2-methyl-2-(2-(1-methyl-3-(4-(trifluoromethoxy)phe...)
Affinity DataEC50:  2.85E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227697(2-(2-(1-ethyl-3-(2-methyl-4-(trifluoromethoxy)phen...)
Affinity DataEC50:  598nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227669((R)-2-(2-(1-ethyl-3-(4-(trifluoromethoxy)phenyl)ur...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at PPARgamma expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227706(2-(2-(1-heptyl-3-(3-(trifluoromethyl)phenyl)ureido...)
Affinity DataEC50:  2.73E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at PPARgamma expressed in HEK293 cells assessed as aP2 gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227704(2-methyl-2-(2-(1-pentyl-3-(4-(trifluoromethylthio)...)
Affinity DataEC50:  46nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227705((R)-2-(2-(1-heptyl-3-(4-(trifluoromethoxy)phenyl)u...)
Affinity DataEC50:  169nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227702(2-(2-(3-(3-bromo-4-(trifluoromethoxy)phenyl)-1-eth...)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227708(2-(2-(3-(3-chloro-4-(trifluoromethoxy)phenyl)-1-et...)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227703(2-(2-(1-heptyl-3-(4-(trifluoromethylthio)phenyl)ur...)
Affinity DataEC50:  229nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227707(2-(2-(1-heptyl-3-phenylureido)-2,3-dihydro-1H-inde...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227669((R)-2-(2-(1-ethyl-3-(4-(trifluoromethoxy)phenyl)ur...)
Affinity DataEC50:  170nMAssay Description:Agonist activity at PPARalpha expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227658(2-(2-(3-(4-(dimethylamino)phenyl)-1-pentylureido)-...)
Affinity DataEC50:  141nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227669((R)-2-(2-(1-ethyl-3-(4-(trifluoromethoxy)phenyl)ur...)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at PPARdelta expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227668(2-methyl-2-(2-(1-propyl-3-(4-(trifluoromethoxy)phe...)
Affinity DataEC50:  158nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227667(2-(2-(3-(3-chlorophenyl)-1-heptylureido)-2,3-dihyd...)
Affinity DataEC50:  2.09E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227666(2-(2-(1-butyl-3-(4-(trifluoromethylthio)phenyl)ure...)
Affinity DataEC50:  160nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227665(2-(2-(3-(3-fluorophenyl)-1-heptylureido)-2,3-dihyd...)
Affinity DataEC50:  2.67E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227664(2-(2-(1-ethyl-3-(4-(trifluoromethoxy)phenyl)ureido...)
Affinity DataEC50:  33nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227663(2-methyl-2-(2-(1-pentyl-3-(4-(trifluoromethoxy)phe...)
Affinity DataEC50:  105nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227659(2-(2-(3-(4-isopropylphenyl)-1-pentylureido)-2,3-di...)
Affinity DataEC50:  159nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227672(2-(2-(1-ethyl-3-methyl-3-(4-(trifluoromethoxy)phen...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227660((R)-2-methyl-2-(2-(3-(4-(trifluoromethoxy)phenyl)u...)
Affinity DataEC50:  146nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227662(2-(2-(3-(4-(dimethylamino)phenyl)-1-heptylureido)-...)
Affinity DataEC50:  252nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227661(2-(2-(1-butyl-3-(4-(trifluoromethoxy)phenyl)ureido...)
Affinity DataEC50:  195nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227657(2-(2-(1-heptyl-3-(4-(methylthio)phenyl)ureido)-2,3...)
Affinity DataEC50:  210nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227656(2-(2-(1-ethyl-3-(4-isopropylphenyl)ureido)-2,3-dih...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM28799(2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)a...)
Affinity DataEC50:  450nMAssay Description:Agonist activity at PPARalpha expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227655(2-(2-(1-heptyl-3-o-tolylureido)-2,3-dihydro-1H-ind...)
Affinity DataEC50:  7.54E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 66 total ) | Next | Last >>
Jump to: