Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50021720
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227151(2-(5-(3-(3-benzyl-8-(trifluoromethyl)quinolin-4-yl...)
Affinity DataEC50:  685nMAssay Description:Agonist activity at human LXRalpha expressed in Huh7 cells by Gal4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227151(2-(5-(3-(3-benzyl-8-(trifluoromethyl)quinolin-4-yl...)
Affinity DataEC50:  84nMAssay Description:Agonist activity at human recombinant PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227151(2-(5-(3-(3-benzyl-8-(trifluoromethyl)quinolin-4-yl...)
Affinity DataEC50:  355nMAssay Description:Agonist activity at human LXRbeta expressed in Huh7 cells by Gal4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataEC50:  178nMAssay Description:Agonist activity at human LXRbeta expressed in Huh7 cells by Gal4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227145(2-(5-((3-(3-methyl-8-(trifluoromethyl)quinolin-4-y...)
Affinity DataEC50:  4.17E+3nMAssay Description:Agonist activity at human LXRbeta expressed in Huh7 cells by Gal4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227147(2-(5-((3-(8-(trifluoromethyl)quinolin-4-yl)phenyl)...)
Affinity DataEC50:  622nMAssay Description:Agonist activity at human LXRbeta expressed in Huh7 cells by Gal4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227145(2-(5-((3-(3-methyl-8-(trifluoromethyl)quinolin-4-y...)
Affinity DataEC50:  7.87E+3nMAssay Description:Agonist activity at human LXRalpha expressed in Huh7 cells by Gal4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM20000(CHEMBL214719 | 2-(4-{3-[3-benzyl-8-(trifluoromethy...)
Affinity DataEC50:  680nMAssay Description:Agonist activity at human recombinant PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227145(2-(5-((3-(3-methyl-8-(trifluoromethyl)quinolin-4-y...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human recombinant PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM20000(CHEMBL214719 | 2-(4-{3-[3-benzyl-8-(trifluoromethy...)
Affinity DataEC50:  240nMAssay Description:Agonist activity at human LXRalpha expressed in Huh7 cells by Gal4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM20000(CHEMBL214719 | 2-(4-{3-[3-benzyl-8-(trifluoromethy...)
Affinity DataEC50:  90nMAssay Description:Agonist activity at human LXRbeta expressed in Huh7 cells by Gal4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227147(2-(5-((3-(8-(trifluoromethyl)quinolin-4-yl)phenyl)...)
Affinity DataEC50:  69nMAssay Description:Agonist activity at human recombinant PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataEC50:  135nMAssay Description:Agonist activity at human LXRalpha expressed in Huh7 cells by Gal4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227147(2-(5-((3-(8-(trifluoromethyl)quinolin-4-yl)phenyl)...)
Affinity DataEC50:  1.19E+3nMAssay Description:Agonist activity at human LXRalpha expressed in Huh7 cells by Gal4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227146(2-(4-(3-(3-benzyl-8-(trifluoromethyl)quinolin-4-yl...)
Affinity DataIC50: 2nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227157(2-(4-((3-(3-benzoyl-8-(trifluoromethyl)quinolin-5-...)
Affinity DataIC50: 2nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227163(2-(4-((3-(3-benzoyl-8-(trifluoromethyl)quinolin-5-...)
Affinity DataIC50: 2nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227161(2-(4-(3-(3-benzyl-8-(trifluoromethyl)quinolin-4-yl...)
Affinity DataIC50: 2nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM20000(CHEMBL214719 | 2-(4-{3-[3-benzyl-8-(trifluoromethy...)
Affinity DataIC50: 2nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227156(2-(4-((3-(3-benzyl-8-(trifluoromethyl)quinolin-4-y...)
Affinity DataIC50: 3nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227159(2-(4-(3-(3-benzyl-8-(trifluoromethyl)quinolin-4-yl...)
Affinity DataIC50: 4nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227158(2-(4-(3-(3-benzyl-8-(trifluoromethyl)quinolin-4-yl...)
Affinity DataIC50: 4nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227162(2-(4-((3-(3-benzoyl-8-(trifluoromethyl)quinolin-5-...)
Affinity DataIC50: 5nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227151(2-(5-(3-(3-benzyl-8-(trifluoromethyl)quinolin-4-yl...)
Affinity DataIC50: 5nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227160(2-(4-((3-(3-benzoyl-8-(trifluoromethyl)quinolin-5-...)
Affinity DataIC50: 5nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227163(2-(4-((3-(3-benzoyl-8-(trifluoromethyl)quinolin-5-...)
Affinity DataIC50: 6nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM20002(CHEMBL216645 | 2-{4-[({3-[3-benzyl-8-(trifluoromet...)
Affinity DataIC50: 7nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataIC50: 9nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM20000(CHEMBL214719 | 2-(4-{3-[3-benzyl-8-(trifluoromethy...)
Affinity DataIC50: 10nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227145(2-(5-((3-(3-methyl-8-(trifluoromethyl)quinolin-4-y...)
Affinity DataIC50: 10nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227154(2-(4-((3-(3-benzoyl-8-(trifluoromethyl)quinolin-5-...)
Affinity DataIC50: 10nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227152(2-(5-(3-(3-benzyl-8-(trifluoromethyl)quinolin-4-yl...)
Affinity DataIC50: 11nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227156(2-(4-((3-(3-benzyl-8-(trifluoromethyl)quinolin-4-y...)
Affinity DataIC50: 11nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataIC50: 13nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227147(2-(5-((3-(8-(trifluoromethyl)quinolin-4-yl)phenyl)...)
Affinity DataIC50: 15nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227160(2-(4-((3-(3-benzoyl-8-(trifluoromethyl)quinolin-5-...)
Affinity DataIC50: 16nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227162(2-(4-((3-(3-benzoyl-8-(trifluoromethyl)quinolin-5-...)
Affinity DataIC50: 17nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227146(2-(4-(3-(3-benzyl-8-(trifluoromethyl)quinolin-4-yl...)
Affinity DataIC50: 21nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227154(2-(4-((3-(3-benzoyl-8-(trifluoromethyl)quinolin-5-...)
Affinity DataIC50: 21nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227161(2-(4-(3-(3-benzyl-8-(trifluoromethyl)quinolin-4-yl...)
Affinity DataIC50: 21nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227157(2-(4-((3-(3-benzoyl-8-(trifluoromethyl)quinolin-5-...)
Affinity DataIC50: 26nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227158(2-(4-(3-(3-benzyl-8-(trifluoromethyl)quinolin-4-yl...)
Affinity DataIC50: 31nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227148(5-(3-(3-benzyl-8-(trifluoromethyl)quinolin-4-yl)be...)
Affinity DataIC50: 35nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM20002(CHEMBL216645 | 2-{4-[({3-[3-benzyl-8-(trifluoromet...)
Affinity DataIC50: 47nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227159(2-(4-(3-(3-benzyl-8-(trifluoromethyl)quinolin-4-yl...)
Affinity DataIC50: 58nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227150(2-(4-((3-(3-benzoyl-8-(trifluoromethyl)quinolin-5-...)
Affinity DataIC50: 65nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227153(2-(4-((3-(3-benzoyl-8-(trifluoromethyl)quinolin-5-...)
Affinity DataIC50: 67nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227150(2-(4-((3-(3-benzoyl-8-(trifluoromethyl)quinolin-5-...)
Affinity DataIC50: 81nMAssay Description:Binding affinity at human LXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227153(2-(4-((3-(3-benzoyl-8-(trifluoromethyl)quinolin-5-...)
Affinity DataIC50: 112nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50227151(2-(5-(3-(3-benzyl-8-(trifluoromethyl)quinolin-4-yl...)
Affinity DataIC50: 123nMAssay Description:Binding affinity at human LXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
Displayed 1 to 50 (of 58 total ) | Next | Last >>
Jump to: